Per Arvidsson

Open for collaboration: an academic platform for drug discovery and development at SciLifeLab

Arvidsson, Per I.; Sandberg, Kristian; Forsberg-Nilsson, Karin

Ingår i Drug Discovery Today, s. 1690-1698, 2016

• DOI för Open for collaboration: an academic platform for drug discovery and development at SciLifeLab
• Ladda ner fulltext (pdf) av Open for collaboration: an academic platform for drug discovery and development at SciLifeLab

Öppenheten förstör chansen till patent

Arvidsson, Per I.; Domeij, Bengt; Hansson, Mats G.; Landegren, Ulf et al.

Ingår i Svenska dagbladet, 2015

Organocatalytic asymmetric cross-aldol reaction of 2-chloroethoxy acetaldehyde: diversity-oriented synthesis of chiral substituted 1,4-dioxanes and morpholines

Sawant, Rajiv T.; Stevenson, Joanne; Odell, Luke R.; Arvidsson, Per I.

Ingår i Tetrahedron, s. 134-141, 2013

• DOI för Organocatalytic asymmetric cross-aldol reaction of 2-chloroethoxy acetaldehyde: diversity-oriented synthesis of chiral substituted 1,4-dioxanes and morpholines

Synthesis of Novel Aryl and Heteroaryl Acyl Sulfonimidamides via Pd-Catalyzed Carbonylation Using a Nongaseous Precursor

Borhade, Sanjay R.; Sandström, Anja; Arvidsson, Per I.

Ingår i Organic Letters, s. 1056-1059, 2013

• DOI för Synthesis of Novel Aryl and Heteroaryl Acyl Sulfonimidamides via Pd-Catalyzed Carbonylation Using a Nongaseous Precursor

Synthesis, 2D-NMR and molecular modelling studies of pentacycloundecane lactam-peptides and peptoids as potential HIV-1 wild type C-SA protease inhibitors

Makatini, Maya M.; Petzold, Katja; Alves, Claudio Nahum; Arvidsson, Per I. et al.

Ingår i Journal of enzyme inhibition and medicinal chemistry (Print), s. 78-88, 2013

• DOI för Synthesis, 2D-NMR and molecular modelling studies of pentacycloundecane lactam-peptides and peptoids as potential HIV-1 wild type C-SA protease inhibitors

Öppenheten förstör chansen till patent

Arvidsson, Per I.; Domeij, Bengt; Hansson, Mats G.; Landegren, Ulf et al.

Ingår i Svenska dagbladet, 2015

Organocatalytic asymmetric cross-aldol reaction of 2-chloroethoxy acetaldehyde: diversity-oriented synthesis of chiral substituted 1,4-dioxanes and morpholines

Sawant, Rajiv T.; Stevenson, Joanne; Odell, Luke R.; Arvidsson, Per I.

Ingår i Tetrahedron, s. 134-141, 2013

• DOI för Organocatalytic asymmetric cross-aldol reaction of 2-chloroethoxy acetaldehyde: diversity-oriented synthesis of chiral substituted 1,4-dioxanes and morpholines

Synthesis of Novel Aryl and Heteroaryl Acyl Sulfonimidamides via Pd-Catalyzed Carbonylation Using a Nongaseous Precursor

Borhade, Sanjay R.; Sandström, Anja; Arvidsson, Per I.

Ingår i Organic Letters, s. 1056-1059, 2013

• DOI för Synthesis of Novel Aryl and Heteroaryl Acyl Sulfonimidamides via Pd-Catalyzed Carbonylation Using a Nongaseous Precursor

Synthesis, 2D-NMR and molecular modelling studies of pentacycloundecane lactam-peptides and peptoids as potential HIV-1 wild type C-SA protease inhibitors

Makatini, Maya M.; Petzold, Katja; Alves, Claudio Nahum; Arvidsson, Per I. et al.

Ingår i Journal of enzyme inhibition and medicinal chemistry (Print), s. 78-88, 2013

• DOI för Synthesis, 2D-NMR and molecular modelling studies of pentacycloundecane lactam-peptides and peptoids as potential HIV-1 wild type C-SA protease inhibitors

Triazolopyrimidinones as gamma-secretase modulators: structure-activity relationship, modulator profile, and in vivo profiling

Yngve, Ulrika; Paulsen, Kim; Macsari, Istvan; Sundstrom, Marie et al.

Ingår i MedChemComm, s. 422-431, 2013

• DOI för Triazolopyrimidinones as gamma-secretase modulators: structure-activity relationship, modulator profile, and in vivo profiling

Sulfonimidamides as Sulfonamides Bioisosteres: Rational Evaluation through Synthetic, in Vitro, and in Vivo Studies with γ-Secretase Inhibitors

Sehgelmeble, Fernando; Jansson, Juliette; Ray, Colin; Rosqvist, Susanne et al.

Ingår i ChemMedChem, s. 396-399, 2012

• DOI för Sulfonimidamides as Sulfonamides Bioisosteres: Rational Evaluation through Synthetic, in Vitro, and in Vivo Studies with γ-Secretase Inhibitors

Imidazopyridine-based inhibitors of glycogen synthase kinase 3: synthesis and evaluation of amide isostere replacements of the carboxamide scaffold

Yngve, Ulrika; Söderman, Peter; Svensson, Mats; Rosqvist, Susanne et al.

Ingår i Chemistry and Biodiversity, s. 2442-2452, 2012

• DOI för Imidazopyridine-based inhibitors of glycogen synthase kinase 3: synthesis and evaluation of amide isostere replacements of the carboxamide scaffold

Asymmetric conjugate addition of thioglycolate to a range of chalcones using tetrahydroisoquinoline (TIQ) N,N '-dioxide ligands

Chakka, Sai Kumar; Francis, Vivian; Cele, Zamani E. D.; Sosibo, Sphelele C. et al.

Ingår i Tetrahedron, s. 616-622, 2012

• DOI för Asymmetric conjugate addition of thioglycolate to a range of chalcones using tetrahydroisoquinoline (TIQ) N,N '-dioxide ligands

Interaction of beta-Amyloid Interactions with Peptide Functionalized Gold Nanoparticles

Hemmaragala, Nanjundaswamy M.; Arvidsson, Per I.; Maguire, Glenn E. M.; Kruger, Hendrik G. et al.

Ingår i Journal of Nanoscience and Nanotechnology, s. 2179-2184, 2012

• DOI för Interaction of beta-Amyloid Interactions with Peptide Functionalized Gold Nanoparticles

Novel bioactivation mechanism of reactive metabolite formation from phenyl methyl-isoxazoles

Bylund, Johan; Macsari, Istvan; Besidski, Yevgeni; Olofsson, Susanne et al.

Ingår i Drug Metabolism And Disposition, s. 2185-2191, 2012

• DOI för Novel bioactivation mechanism of reactive metabolite formation from phenyl methyl-isoxazoles

3-Oxoisoindoline-1-carboxamides: Potent, State-Dependent Blockers of Voltage-Gated Sodium Channel Na(V)1.7 with Efficacy in Rat Pain Models

Macsari, Istvan; Besidski, Yeygeni; Csjernyik, Gabor; Nilsson, Linda I. et al.

Ingår i Journal of Medicinal Chemistry, s. 6866-6880, 2012

• DOI för 3-Oxoisoindoline-1-carboxamides: Potent, State-Dependent Blockers of Voltage-Gated Sodium Channel Na(V)1.7 with Efficacy in Rat Pain Models

Microwave-Assisted Synthesis of Guanidine Organocatalysts Bearing a Tetrahydroisoquinoline Framework and Their Evaluation in Michael Addition Reactions

Naicker, Tricia; Arvidsson, Per I.; Kruger, Hendrik G.; Maguire, Glenn E. M. et al.

Ingår i European Journal of Organic Chemistry, s. 3331-3337, 2012

• DOI för Microwave-Assisted Synthesis of Guanidine Organocatalysts Bearing a Tetrahydroisoquinoline Framework and Their Evaluation in Michael Addition Reactions

Synthesis and arylation of unprotected sulfonimidamides

Maldonado, Matias Funes; Sehgelmeble, Fernando; Bjarnemark, Fanny; Svensson, Mats et al.

Ingår i Tetrahedron, s. 7456-7462, 2012

• DOI för Synthesis and arylation of unprotected sulfonimidamides

Alzheimer's Disease: Presenilin 2-Sparing γ-Secretase Inhibition Is a Tolerable Aβ Peptide-Lowering Strategy

Borgegård, Tomas; Gustavsson, Susanne; Nilsson, Charlotte; Parpal, Santiago et al.

Ingår i Journal of Neuroscience, s. 17297-17305, 2012

• DOI för Alzheimer's Disease: Presenilin 2-Sparing γ-Secretase Inhibition Is a Tolerable Aβ Peptide-Lowering Strategy

Pentacycloundecane-diol-Based HIV-1 Protease Inhibitors: Biological Screening, 2D NMR, and Molecular Simulation Studies

Honarparvar, Bahareh; Makatini, Maya M.; Pawar, Sachin A.; Petzold, Katja et al.

Ingår i ChemMedChem, s. 1009-1019, 2012

• DOI för Pentacycloundecane-diol-Based HIV-1 Protease Inhibitors: Biological Screening, 2D NMR, and Molecular Simulation Studies

Synthesis, screening and computational investigation of pentacycloundecane-peptoids as potent CSA-HIV PR inhibitors

Makatini, Maya M.; Petzold, Katja; Arvidsson, Per I.; Honarparvar, Bahareh et al.

Ingår i European Journal of Medicinal Chemistry, s. 459-467, 2012

• DOI för Synthesis, screening and computational investigation of pentacycloundecane-peptoids as potent CSA-HIV PR inhibitors

Phenyl isoxazole voltage-gated sodium channel blockers: structure and activity relationship

Macsari, Istvan; Sandberg, Lars; Besidski, Yevgeni; Gravenfors, Ylva et al.

Ingår i Bioorganic & Medicinal Chemistry Letters, s. 3871-3876, 2011

• DOI för Phenyl isoxazole voltage-gated sodium channel blockers: structure and activity relationship

Pentacycloundecane-based inhibitors of wild-type C-South African HIV-protease

Makatini, Maya M.; Petzold, Katja; Sriharsha, Shimoga N.; Soliman, Mahmoud E. S. et al.

Ingår i Bioorganic & Medicinal Chemistry Letters, s. 2274-2277, 2011

• DOI för Pentacycloundecane-based inhibitors of wild-type C-South African HIV-protease

Synthesis and structural studies of pentacycloundecane-based HIV-1 PR inhibitors: A hybrid 2D NMR and docking/QM/MM/MD approach

Makatini, Maya M.; Petzold, Katja; Sriharsha, Shimoga N.; Ndlovu, N. et al.

Ingår i European Journal of Medicinal Chemistry, s. 3976-3985, 2011

• DOI för Synthesis and structural studies of pentacycloundecane-based HIV-1 PR inhibitors: A hybrid 2D NMR and docking/QM/MM/MD approach

Tetrahydroisoquinoline-Based N-Oxides as Chiral Organocatalysts for the Asymmetric Allylation of Aldehydes

Naicker, Tricia; Arvidsson, Per I; Kruger, Hendrik G; Maguire, Glenn E M et al.

Ingår i European Journal of Organic Chemistry, s. 6923-6932, 2011

• DOI för Tetrahydroisoquinoline-Based N-Oxides as Chiral Organocatalysts for the Asymmetric Allylation of Aldehydes

Design and study of peptide-based inhibitors of amylin cytotoxicity

Muthusamy, Karen; Arvidsson, Per I.; Govender, Patrick; Kruger, Hendrik G. et al.

Ingår i Bioorganic & Medicinal Chemistry Letters, s. 1360-1362, 2010

• DOI för Design and study of peptide-based inhibitors of amylin cytotoxicity

Novel tetrahydroisoquinoline based organocatalysts for asymmetric Diels–Alder reactions: insight into the catalytic mode using ROESY NMR and DFT studies

Naicker, Tricia; Petzold, Katja; Singh, Thishana; Arvidsson, Per I. et al.

Ingår i Tetrahedron, s. 2859-2867, 2010

• DOI för Novel tetrahydroisoquinoline based organocatalysts for asymmetric Diels–Alder reactions: insight into the catalytic mode using ROESY NMR and DFT studies

In vitro ADMET and physicochemical investigations of poly-N-methylated peptides designed to inhibit Aβ aggregation

Bose, Partha Pratim; Chatterjee, Urmimala; Hubatsch, Ina; Artursson, Per et al.

Ingår i Bioorganic & Medicinal Chemistry, s. 5896-5902, 2010

• DOI för In vitro ADMET and physicochemical investigations of poly-N-methylated peptides designed to inhibit Aβ aggregation

Effects of Congo Red on A beta(1-40) Fibril Formation Process and Morphology

Bose, Partha Pratim; Chatterjee, Urmimala; Xie, Ling; Johansson, Jan et al.

Ingår i ACS CHEMICAL NEUROSCIENCE, s. 315-324, 2010

• DOI för Effects of Congo Red on A beta(1-40) Fibril Formation Process and Morphology

Microwave Assisted SPPS of Amylin and Its Toxicity of the Pure Product to RIN-5F Cells

Muthusamy, Karen; Albericio, Fernando; Arvidsson, Per I.; Govender, Patrick et al.

Ingår i Biopolymers, s. 323-330, 2010

• DOI för Microwave Assisted SPPS of Amylin and Its Toxicity of the Pure Product to RIN-5F Cells

Synthesis and NMR elucidation of novel pentacycloundecane-based peptides

Altaib, Mohamed S.; Arvidsson, Per I.; Govender, Thavendran; Maguire, Glenn E. M. et al.

Ingår i Magnetic Resonance in Chemistry, s. 435-442, 2010

• DOI för Synthesis and NMR elucidation of novel pentacycloundecane-based peptides

Poly-N-methylated Amyloid β-Peptide (Aβ) C-Terminal Fragments Reduce Aβ Toxicity in Vitro and in Drosophila melanogaster

Pratim Bose, Partha; Chatterjee, Urmimala; Nerelius, Charlotte; Govender, Thavendran et al.

Ingår i Journal of Medicinal Chemistry, s. 8002-8009, 2009

• DOI för Poly-N-methylated Amyloid β-Peptide (Aβ) C-Terminal Fragments Reduce Aβ Toxicity in Vitro and in Drosophila melanogaster

Application of (S,S)-Pentacycloundecane bis(4-Phenyloxazoline) as a Novel Chiral Ligand for Catalysis of the Asymmetric Diels-Alder Reaction of Cyclopentadiene with 3-Acryloyl-2-oxazolidinone

Arvidsson, Per I.; Govender, Thavendran; Kruger, G; Maguire, M et al.

Ingår i South African Journal of Chemistry, s. 60-U78, 2009

Synthesis and application of novel imidazole and 1H-tetrazolic acid containing catalysts in enantioselective organocatalyzed Diels-Alder reactions

Hartikka, Antti; Hojabri, Leila; Bose, Pratim; Arvidsson, Per I.

Ingår i Tetrahedron, s. 1871-1876, 2009

• DOI för Synthesis and application of novel imidazole and 1H-tetrazolic acid containing catalysts in enantioselective organocatalyzed Diels-Alder reactions

Cobalt-doped beta-peptide nanotubes: A class of spintronic materials

Sanyal, Biplab; Eriksson, Olle; Arvidsson, Per I.

Ingår i Physical Review B. Condensed Matter and Materials Physics, s. 155407, 2008

• DOI för Cobalt-doped beta-peptide nanotubes: A class of spintronic materials

Design and synthesis of glycosylated b 3-peptides capable of folding into the 314-helical conformation in water

Norgren, Anna S.; Arvidsson, Per I.

Ingår i Journal of Organic Chemistry, s. 5272-5278, 2008

• DOI för Design and synthesis of glycosylated b 3-peptides capable of folding into the 314-helical conformation in water

Facile synthesis of N-protected amino acid assisted by microwave irradiation

Zhang, Suode; Arvidsson, Per I.

Ingår i International journal of peptide research and therapeutics, s. 219-222, 2008

• DOI för Facile synthesis of N-protected amino acid assisted by microwave irradiation

Beta- and gamma-di- and tripeptides as potential substrates for the oligopeptide transporter hPepT1

Hubatsch, Ina; Arvidsson, Per I.; Seebach, Dieter; Luthman, Kristina et al.

Ingår i Journal of Medicinal Chemistry, s. 5238-5242, 2007

• DOI för Beta- and gamma-di- and tripeptides as potential substrates for the oligopeptide transporter hPepT1

A new Imidazole-Containing Imidazolidinone Catalyst for Organocatalyzed Asymmetric Conjugate Addition of Nitroalkanes to Aldehydes

Hojabri, Leila; Hartikka, Antti; Moghaddam, Firouz. M; Arvidsson, Per I.

Ingår i Advanced Synthesis and Catalysis, s. 740-748, 2007

• DOI för A new Imidazole-Containing Imidazolidinone Catalyst for Organocatalyzed Asymmetric Conjugate Addition of Nitroalkanes to Aldehydes

Tetrazolic Acid Functionalized Dihydroindol: Rational Design of a Highly Selective Cyclopropanation Organocatalyst

Hartikka, Antti; Arvidsson, Per. I

Ingår i Journal of Organic Chemistry, s. 5874-5877, 2007

• DOI för Tetrazolic Acid Functionalized Dihydroindol: Rational Design of a Highly Selective Cyclopropanation Organocatalyst

Glycosylated Foldamers: Synthesis of Carbohydrate-modified β3hSer and Incorporation into β-Peptides

Norgren, Anna S.; Norberg, Thomas; Arvidsson, Per I.

Ingår i Journal of Peptide Science, s. 717-727, 2007

• DOI för Glycosylated Foldamers: Synthesis of Carbohydrate-modified β3hSer and Incorporation into β-Peptides

Biomolecular Recognition of Glycosylated β3-Peptides by GalNAc Specific Lectins

Norgren, Anna S.; Geitmann, Matthis; Danielson, U. Helena; Arvidsson, Per I.

Ingår i Journal of Molecular Recognition, s. 132-138, 2007

• DOI för Biomolecular Recognition of Glycosylated β3-Peptides by GalNAc Specific Lectins

Application of novel sulfonamides in enantioselective organocatalyzed cyclopropanation

Hartikka, Antti; Slosarczyk, Adam; Arvidsson, Per

Ingår i Tetrahedron, s. 1403-1409, 2007

• DOI för Application of novel sulfonamides in enantioselective organocatalyzed cyclopropanation

Synthesis and circular dichroism spectroscopic investigations of oligomeric β-peptoids with α-chiral side chains

Norgren, Anna; Zhang, Suode; Arvidsson, Per

Ingår i Organic Letters, s. 4533-4536, 2006

• DOI för Synthesis and circular dichroism spectroscopic investigations of oligomeric β-peptoids with α-chiral side chains

Mechanistic Insights into the Phosphine-Free RuCp*-Diamine-Catalyzed Hydrogenation of Aryl Ketones: Experimental and Theoretical Evidence for an Alcohol-Mediated Dihydrogen Activation

Hedberg, Christian; Källström, Klas; Arvidsson, Per; Brandt, Peter et al.

Ingår i J. Am. Chem. Soc., s. 15083-15090, 2005

• DOI för Mechanistic Insights into the Phosphine-Free RuCp*-Diamine-Catalyzed Hydrogenation of Aryl Ketones: Experimental and Theoretical Evidence for an Alcohol-Mediated Dihydrogen Activation

Exploring the Antibacterial and Hemolytic Activity of Shorter- and Longer-Chain B-, a,B-, and y-Peptides, and of B-Peptides from B2-3-Aza- and B3-2-Methylidene-amino Acids Bearing Proteinogenic Side Chains - A Survey

Arvidsson, Per; Ryder, Neil S.; Weiss, H. Markus; Hook, David F. et al.

Ingår i Chemistry & Biodiversity, s. 401-420, 2005

An Improved Synthesis of Fmoc-N-methyl-a-amino Acids

Zhang, Suode; Govender, Thavendran; Norström, Thomas; Arvidsson, Per

Ingår i J. Org. Chem., s. 6918-6920, 2005

Cyclic B-Tetra- and Pentapeptides: Synthesis through On-Resin Cyclization and Confomrational Studies by X-Ray, NMR and CD Spectroscopy and Theoretical Calculations

Buttner, Frank; Norgren, Anna; Zhang, Suode; Prabpai, Samran et al.

Ingår i Chem. Eur. J., s. 6145-6158, 2005

• DOI för Cyclic B-Tetra- and Pentapeptides: Synthesis through On-Resin Cyclization and Confomrational Studies by X-Ray, NMR and CD Spectroscopy and Theoretical Calculations

cyclo(ß-Asp-ß3-hVal-ß3-hLys)-Solid-Phase Synthesis and Solution Structure of a Water Soluble ß-Tripeptide

Büttner, Frank; Erdélyi, Máté; Arvidsson, Per

Ingår i Helvetica Chimica Acta, s. 2735-2741, 2004

Rational design of asymmetric organocatalysts-increased reactivity and solvent scope with a tetrazolic acid

Hartikka, Antti; Arvidsson, Per

Ingår i Tetrahedron Asymmetry, s. 1831-1834, 2004

Syntheses an CD-Spectroscopic Investigations of Longer-Chain B-Peptides: Preparation by Solid-Phase Couplings of Single Amino Acids, Dipeptides, and Tripeptides

Arvidsson, Per; Frackenpohl, J; Seebach, D

Ingår i Helvetica Chemica Acta, s. 1552-1553, 2003

Antibiotic and Hemolytic Activity of a B2/B3 Peptide Capable of Folding into a 12/10-Helical Secondary Structure

Arvidsson, Per; Ryder, N; Weiss, M; Gross, G et al.

Ingår i ChemBioChem, s. 1345-1347, 2003

Open for collaboration: an academic platform for drug discovery and development at SciLifeLab

Arvidsson, Per I.; Sandberg, Kristian; Forsberg-Nilsson, Karin

Ingår i Drug Discovery Today, s. 1690-1698, 2016

• DOI för Open for collaboration: an academic platform for drug discovery and development at SciLifeLab
• Ladda ner fulltext (pdf) av Open for collaboration: an academic platform for drug discovery and development at SciLifeLab