Luke Odell

Spatial visualization of comprehensive brain neurotransmitter systems and neuroactive substances by selective in situ chemical derivatization mass spectrometry imaging

Shariatgorji, Reza; Nilsson, Anna; Fridjonsdottir, Elva; Strittmatter, Nicole et al.

Ingår i Nature Protocols, s. 3298-3321, 2021

• DOI för Spatial visualization of comprehensive brain neurotransmitter systems and neuroactive substances by selective in situ chemical derivatization mass spectrometry imaging

The Wittig Bioconjugation of Maleimide Derived, Water Soluble Phosphonium Ylides to Aldehyde-Tagged Proteins

Hartmann, Rafael W.; Pijnappel, Matthijs; Nilvebrant, Johan; Helgudottir, Hildur Run et al.

Ingår i Organic and biomolecular chemistry, s. 10417-10423, 2021

• DOI för The Wittig Bioconjugation of Maleimide Derived, Water Soluble Phosphonium Ylides to Aldehyde-Tagged Proteins
• Ladda ner fulltext (pdf) av The Wittig Bioconjugation of Maleimide Derived, Water Soluble Phosphonium Ylides to Aldehyde-Tagged Proteins

Sustainability in drug discovery

Wynendaele, Evelien; Furman, Christophe; Wielgomas, Bartosz; Larsson, Per et al.

Ingår i Medicine in Drug Discovery, 2021

• DOI för Sustainability in drug discovery
• Ladda ner fulltext (pdf) av Sustainability in drug discovery

Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.

Hartmann, Rafael; Fahrner, Raphael; Shevshenko, Denys; Fryknäs, Mårten et al.

Ingår i ChemMedChem, s. 2500-2512, 2020

• DOI för Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.
• Ladda ner fulltext (pdf) av Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.

Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF₃⦁SMe₂

Söderström, Marcus; Zamaratski, Edouard; Odell, Luke R.

Ingår i European Journal of Organic Chemistry, s. 5402-5408, 2019

• DOI för Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF₃⦁SMe₂
• Ladda ner fulltext (pdf) av Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF₃⦁SMe₂

Synthesis and preclinical evaluation of the CRTH2 antagonist [¹¹C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

Eriksson, Jonas; Roy, Tamal; Sawadjoon, Supaporn; Bachmann, Kim et al.

Ingår i Nuclear Medicine and Biology, s. 1-10, 2019

• DOI för Synthesis and preclinical evaluation of the CRTH2 antagonist [¹¹C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass
• Ladda ner fulltext (pdf) av Synthesis and preclinical evaluation of the CRTH2 antagonist [¹¹C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

Comprehensive mapping of neurotransmitter networks by MALDI-MS imaging

Shariatgorji, Mohammadreza; Nilsson, Anna; Fridjonsdottir, Elva; Vallianatou, Theodosia et al.

Ingår i Nature Methods, s. 1021-1028, 2019

• DOI för Comprehensive mapping of neurotransmitter networks by MALDI-MS imaging

Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

Schembri, Luke S; Eriksson, Jonas; Odell, Luke R.

Ingår i Journal of Organic Chemistry, s. 6970-6981, 2019

• DOI för Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

Palladium-mediated C-11-carbonylations using aryl halides and cyanamide

Nordeman, Patrik; Chow, Shiao Y.; Odell, A. F.; Antoni, Gunnar et al.

Ingår i Organic and biomolecular chemistry, s. 4875-4881, 2017

• DOI för Palladium-mediated C-11-carbonylations using aryl halides and cyanamide

Synthesis of N-Sulfonyl Amidines and Acyl Sulfonyl Ureas from Sulfonyl Azides, Carbon Monoxide, and Amides

Chow, Shiao Y.; Odell, Luke R.

Ingår i Journal of Organic Chemistry, s. 2515-2522, 2017

• DOI för Synthesis of N-Sulfonyl Amidines and Acyl Sulfonyl Ureas from Sulfonyl Azides, Carbon Monoxide, and Amides

Acetic acid-promoted cascade N-acyliminium ion/aza-Prins cyclization: stereoselective synthesis of functionalized fused tricyclic piperidines

Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

Ingår i Chemical Communications, s. 2110-2113, 2017

• DOI för Acetic acid-promoted cascade N-acyliminium ion/aza-Prins cyclization: stereoselective synthesis of functionalized fused tricyclic piperidines

Palladium and Visible-Light Mediated Carbonylative Suzuki-Miyaura Coupling of Unactivated Alkyl Halides and Aryl Boronic Acids

Roslin, Sara; Odell, Luke R.

Ingår i Chemical Communications, s. 6895-6898, 2017

• DOI för Palladium and Visible-Light Mediated Carbonylative Suzuki-Miyaura Coupling of Unactivated Alkyl Halides and Aryl Boronic Acids

Microwave-Assisted Branching Cascades: A Route to Diverse 3,4-Dihydroquinazolinone-Embedded Polyheterocyclic Scaffolds

Sawant, Rajiv T.; Stevens, Marc Y.; Sköld, Christian; Odell, Luke R.

Ingår i Organic Letters, s. 5392-5395, 2016

• DOI för Microwave-Assisted Branching Cascades: A Route to Diverse 3,4-Dihydroquinazolinone-Embedded Polyheterocyclic Scaffolds

Sulfonyl Azides as Precursors in Ligand-free Palladium-Catalyzed Synthesis of Sulfonyl Carbamates and Sulfonyl Ureas and Synthesis of Sulfonamides

Chow, Shiao; Stevens, Marc; Odell, Luke

Ingår i Journal of Organic Chemistry, s. 2681-2691, 2016

• DOI för Sulfonyl Azides as Precursors in Ligand-free Palladium-Catalyzed Synthesis of Sulfonyl Carbamates and Sulfonyl Ureas and Synthesis of Sulfonamides

Heterocyclic scaffold-fused dimethoxy-dibenzocyclooctynes for photoactivatable click chemistry

Larsson, N. Alfred; Jo, Taegeun; Bremberg, Ulf; Crespi, Stefano et al.

Ingår i Organic and biomolecular chemistry, s. 120-126, 2026

• DOI för Heterocyclic scaffold-fused dimethoxy-dibenzocyclooctynes for photoactivatable click chemistry
• Ladda ner fulltext (pdf) av Heterocyclic scaffold-fused dimethoxy-dibenzocyclooctynes for photoactivatable click chemistry

Late-stage defluorinative functionalization: synthesis of thio-amides and heterocycles from trifluoromethylarenes

Söderström, Marcus; Olaniran Håkansson, Esther; Odell, Luke R.

Ingår i Organic Chemistry Frontiers, s. 1275-1280, 2026

• DOI för Late-stage defluorinative functionalization: synthesis of thio-amides and heterocycles from trifluoromethylarenes
• Ladda ner fulltext (pdf) av Late-stage defluorinative functionalization: synthesis of thio-amides and heterocycles from trifluoromethylarenes

A novel ¹⁸F-labelled tetrazine ester prosthetic group for improved radiolabelling and in vivo stability of proteins and peptides

Lechi, Francesco; Odell, Luke R.; Wegrzyniak, Olivia; Balestri, Lorenzo et al.

Ingår i EJNMMI Radiopharmacy and Chemistry, 2026

• DOI för A novel ¹⁸F-labelled tetrazine ester prosthetic group for improved radiolabelling and in vivo stability of proteins and peptides
• Ladda ner fulltext (pdf) av A novel ¹⁸F-labelled tetrazine ester prosthetic group for improved radiolabelling and in vivo stability of proteins and peptides

Derivatization of Small Molecules using Deuterated Analog of Reactive Matrix to Facilitate Identification in Mass Spectrometry Imaging

Vallianatou, Theodosia; Ilic Balestri, Lorenzo Jacopo; Nilsson, Anna; Zhang, Xiaoqun et al.

Ingår i Chemistry-Methods, 2025

• DOI för Derivatization of Small Molecules using Deuterated Analog of Reactive Matrix to Facilitate Identification in Mass Spectrometry Imaging
• Ladda ner fulltext (pdf) av Derivatization of Small Molecules using Deuterated Analog of Reactive Matrix to Facilitate Identification in Mass Spectrometry Imaging

Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations

Beveridge, Julia; Söderström, Marcus; Balestri, Lorenzo; Prieto-Díaz, Rubén et al.

Ingår i Synlett, s. 2666-2670, 2025

• DOI för Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations
• Ladda ner fulltext (pdf) av Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations

Heterocyclic scaffold-fused dimethoxy-dibenzocyclooctynes for photoactivatable click chemistry

Larsson, N. Alfred; Jo, Taegeun; Bremberg, Ulf; Crespi, Stefano et al.

Ingår i Organic and biomolecular chemistry, s. 120-126, 2026

• DOI för Heterocyclic scaffold-fused dimethoxy-dibenzocyclooctynes for photoactivatable click chemistry
• Ladda ner fulltext (pdf) av Heterocyclic scaffold-fused dimethoxy-dibenzocyclooctynes for photoactivatable click chemistry

Late-stage defluorinative functionalization: synthesis of thio-amides and heterocycles from trifluoromethylarenes

Söderström, Marcus; Olaniran Håkansson, Esther; Odell, Luke R.

Ingår i Organic Chemistry Frontiers, s. 1275-1280, 2026

• DOI för Late-stage defluorinative functionalization: synthesis of thio-amides and heterocycles from trifluoromethylarenes
• Ladda ner fulltext (pdf) av Late-stage defluorinative functionalization: synthesis of thio-amides and heterocycles from trifluoromethylarenes

A novel ¹⁸F-labelled tetrazine ester prosthetic group for improved radiolabelling and in vivo stability of proteins and peptides

Lechi, Francesco; Odell, Luke R.; Wegrzyniak, Olivia; Balestri, Lorenzo et al.

Ingår i EJNMMI Radiopharmacy and Chemistry, 2026

• DOI för A novel ¹⁸F-labelled tetrazine ester prosthetic group for improved radiolabelling and in vivo stability of proteins and peptides
• Ladda ner fulltext (pdf) av A novel ¹⁸F-labelled tetrazine ester prosthetic group for improved radiolabelling and in vivo stability of proteins and peptides

Derivatization of Small Molecules using Deuterated Analog of Reactive Matrix to Facilitate Identification in Mass Spectrometry Imaging

Vallianatou, Theodosia; Ilic Balestri, Lorenzo Jacopo; Nilsson, Anna; Zhang, Xiaoqun et al.

Ingår i Chemistry-Methods, 2025

• DOI för Derivatization of Small Molecules using Deuterated Analog of Reactive Matrix to Facilitate Identification in Mass Spectrometry Imaging
• Ladda ner fulltext (pdf) av Derivatization of Small Molecules using Deuterated Analog of Reactive Matrix to Facilitate Identification in Mass Spectrometry Imaging

Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations

Beveridge, Julia; Söderström, Marcus; Balestri, Lorenzo; Prieto-Díaz, Rubén et al.

Ingår i Synlett, s. 2666-2670, 2025

• DOI för Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations
• Ladda ner fulltext (pdf) av Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations

Pretargeted brain PET imaging reveals amyloid-β pathology using a TCO-modified antibody and a fluorine-18-labeled tetrazine

Lopes van den Broek, Sara; Eriksson, Jonas; Yang, Qiaojun; Bucher, Nadja M. et al.

Ingår i Translational Neurodegeneration, 2025

• DOI för Pretargeted brain PET imaging reveals amyloid-β pathology using a TCO-modified antibody and a fluorine-18-labeled tetrazine
• Ladda ner fulltext (pdf) av Pretargeted brain PET imaging reveals amyloid-β pathology using a TCO-modified antibody and a fluorine-18-labeled tetrazine

Novel Macrocyclic Peptidomimetics Targeting the Insulin-Regulated Aminopeptidase (IRAP): Design, Synthesis and Evaluation

Olaniran Håkansson, Esther; Balestri, Lorenzo Jacopo Ilic; Puthiyaparambath, Sharathna; Moes, Sebastian et al.

Ingår i RSC Medicinal chemistry, s. 5059-5069, 2025

• DOI för Novel Macrocyclic Peptidomimetics Targeting the Insulin-Regulated Aminopeptidase (IRAP): Design, Synthesis and Evaluation
• Ladda ner fulltext (pdf) av Novel Macrocyclic Peptidomimetics Targeting the Insulin-Regulated Aminopeptidase (IRAP): Design, Synthesis and Evaluation

Insulin-regulated aminopeptidase inhibitor C9 restores cellular activity in methadone-damaged primary cell cultures

Stam, Frida; Lind, Sara Florén; Nylander, Erik; Olaniran Håkansson, Esther et al.

Ingår i Neuroscience Letters, 2025

• DOI för Insulin-regulated aminopeptidase inhibitor C9 restores cellular activity in methadone-damaged primary cell cultures
• Ladda ner fulltext (pdf) av Insulin-regulated aminopeptidase inhibitor C9 restores cellular activity in methadone-damaged primary cell cultures

A Multicomponent aza-Prins Strategy for the Diastereoselective Synthesis of Piperidine-Fused Dihydroquinazolinones

Dybeck, Lovisa; Baudoin, Morgane; Odell, Luke R.

Ingår i European Journal of Organic Chemistry, 2025

• DOI för A Multicomponent aza-Prins Strategy for the Diastereoselective Synthesis of Piperidine-Fused Dihydroquinazolinones
• Ladda ner fulltext (pdf) av A Multicomponent aza-Prins Strategy for the Diastereoselective Synthesis of Piperidine-Fused Dihydroquinazolinones

A Diastereoselective Mizoroki-Heck Reaction for Synthesis of Spirooxindole-Based Nonnatural Amino Acids Using a Boc-Protected Amine Chiral Auxiliary

Lindman, Jens; Puthiyaparambath, Sharathna; Gising, Johan; Odell, Luke R. et al.

Ingår i Synlett, s. 2009-2013, 2025

• DOI för A Diastereoselective Mizoroki-Heck Reaction for Synthesis of Spirooxindole-Based Nonnatural Amino Acids Using a Boc-Protected Amine Chiral Auxiliary
• Ladda ner fulltext (pdf) av A Diastereoselective Mizoroki-Heck Reaction for Synthesis of Spirooxindole-Based Nonnatural Amino Acids Using a Boc-Protected Amine Chiral Auxiliary

A preclinical study on the influence of linkers in [⁶⁸Ga]Ga-NOTA-X-RM26 radiotracers for PET imaging of GRPR expression

Olaniran Håkansson, Esther; Zelepukin, Ivan V.; Obeid, Karim; Bitzios, Athanasios et al.

Ingår i EJNMMI Research, 2025

• DOI för A preclinical study on the influence of linkers in [⁶⁸Ga]Ga-NOTA-X-RM26 radiotracers for PET imaging of GRPR expression
• Ladda ner fulltext (pdf) av A preclinical study on the influence of linkers in [⁶⁸Ga]Ga-NOTA-X-RM26 radiotracers for PET imaging of GRPR expression

One-pot, chemoselective desulfurative functionalization of cysteine containing peptides using pyridinium salts

van den Heuvel, Jeroen W.; Olaniran Håkansson, Esther; Skillinghaug, Bobo; Odell, Luke R.

Ingår i Chemical Communications, s. 10347-10350, 2025

• DOI för One-pot, chemoselective desulfurative functionalization of cysteine containing peptides using pyridinium salts
• Ladda ner fulltext (pdf) av One-pot, chemoselective desulfurative functionalization of cysteine containing peptides using pyridinium salts

Synthesis and In Vitro Profiling of Psilocin Derivatives: Improved Stability and Synthetic Properties

Eklund, Julia; Bremberg, Ulf; Larsson, Jessica; Torkelsson, Edvard et al.

Ingår i Journal of Medicinal Chemistry, s. 7153-7165, 2025

• DOI för Synthesis and In Vitro Profiling of Psilocin Derivatives: Improved Stability and Synthetic Properties
• Ladda ner fulltext (pdf) av Synthesis and In Vitro Profiling of Psilocin Derivatives: Improved Stability and Synthetic Properties

Synthesis and preclinical evaluation of gastrin releasing peptide receptor antagonist [¹⁸F]MeTz-PEG2-RM26 for positron emission tomography

Kanellopoulos, Panagiotis; Lundmark, Fanny; Abouzayed, Ayman; Balestri, Lorenzo Jacopo Ilic et al.

Ingår i EJNMMI Radiopharmacy and Chemistry, 2025

• DOI för Synthesis and preclinical evaluation of gastrin releasing peptide receptor antagonist [¹⁸F]MeTz-PEG2-RM26 for positron emission tomography
• Ladda ner fulltext (pdf) av Synthesis and preclinical evaluation of gastrin releasing peptide receptor antagonist [¹⁸F]MeTz-PEG2-RM26 for positron emission tomography

Defluorinative thio-functionalization: direct synthesis of methyl-dithioesters from trifluoromethylarenes

Söderström, Marcus; Olaniran Håkansson, Esther; Odell, Luke R.

Ingår i Chemical Communications, s. 145-148, 2025

• DOI för Defluorinative thio-functionalization: direct synthesis of methyl-dithioesters from trifluoromethylarenes
• Ladda ner fulltext (pdf) av Defluorinative thio-functionalization: direct synthesis of methyl-dithioesters from trifluoromethylarenes

Optimized method for fluorine-18 radiolabeling of Affibody molecules using RESCA

Lechi, Francesco; Eriksson, Jonas; Odell, Luke R.; Wegrzyniak, Olivia et al.

Ingår i EJNMMI Radiopharmacy and Chemistry, 2024

• DOI för Optimized method for fluorine-18 radiolabeling of Affibody molecules using RESCA
• Ladda ner fulltext (pdf) av Optimized method for fluorine-18 radiolabeling of Affibody molecules using RESCA

Inhibition of IRAP Enhances the Expression of Pro-Cognitive Markers Drebrin and MAP2 in Rat Primary Neuronal Cells

Stam, Frida; Lind, Sara Florén; Nylander, Erik; Olaniran, Esther et al.

Ingår i International Journal of Molecular Sciences, 2024

• DOI för Inhibition of IRAP Enhances the Expression of Pro-Cognitive Markers Drebrin and MAP2 in Rat Primary Neuronal Cells
• Ladda ner fulltext (pdf) av Inhibition of IRAP Enhances the Expression of Pro-Cognitive Markers Drebrin and MAP2 in Rat Primary Neuronal Cells

Synthesis of N-Alkenylated Heterocycles via T₃P-Promoted Condensation with Ketones

Balestri, Lorenzo Jacopo Ilic; Beveridge, Julia; Gising, Johan; Odell, Luke R.

Ingår i Journal of Organic Chemistry, s. 11203-11214, 2024

• DOI för Synthesis of N-Alkenylated Heterocycles via T₃P-Promoted Condensation with Ketones
• Ladda ner fulltext (pdf) av Synthesis of N-Alkenylated Heterocycles via T₃P-Promoted Condensation with Ketones

Benzylhydroxamic acids as inhibitors of insulin regulated aminopeptidase (IRAP)

Beveridge, Julia; Söderström, Marcus; Prieto-Díaz, Rubén; Gutierrez-de-Teran, Hugo et al.

Ingår i European Journal of Medicinal Chemistry Reports, 2024

• DOI för Benzylhydroxamic acids as inhibitors of insulin regulated aminopeptidase (IRAP)
• Ladda ner fulltext (pdf) av Benzylhydroxamic acids as inhibitors of insulin regulated aminopeptidase (IRAP)

Hydrazide-based reactive matrices for the sensitive detection of aldehydes and ketones by MALDI mass spectrometry imaging

Lodén, Henrik; Schembri, Luke S; Nilsson, Anna; Kaya, Ibrahim et al.

Ingår i Chemical Communications, s. 9238-9241, 2024

• DOI för Hydrazide-based reactive matrices for the sensitive detection of aldehydes and ketones by MALDI mass spectrometry imaging

Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET

Schlein, Eva; Rokka, Johanna; Odell, Luke R.; Lopes van den Broek, Sara et al.

Ingår i EJNMMI Radiopharmacy and Chemistry, 2024

• DOI för Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
• Ladda ner fulltext (pdf) av Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET

A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane

Schembri, Luke S; Olaniran, Esther; Söderström, Marcus; Skillinghaug, Bobo et al.

Ingår i Advanced Synthesis and Catalysis, s. 1839-1845, 2023

• DOI för A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane
• Ladda ner fulltext (pdf) av A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane

[¹⁸F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44

Cheung, Pierre; Amin, Mohammad A.; Zhang, Bo; Lechi, Francesco et al.

Ingår i Pharmaceutics, 2023

• DOI för [¹⁸F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44
• Ladda ner fulltext (pdf) av [¹⁸F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44

Synthesis of Substituted Indazole Acetic Acids by N-N Bond Forming Reactions

Odell, Luke R.; Skillinghaug, Bobo; Matt, Christof; Wu, Peng et al.

Ingår i European Journal of Organic Chemistry, 2023

• DOI för Synthesis of Substituted Indazole Acetic Acids by N-N Bond Forming Reactions
• Ladda ner fulltext (pdf) av Synthesis of Substituted Indazole Acetic Acids by N-N Bond Forming Reactions

Thioacetalation and Multi-Component Thiomethylative Friedel-Crafts Arylation Using BF₃SMe₂

Söderström, Marcus; Matt, Christof; Odell, Luke R.

Ingår i ACS Omega, s. 4320-4330, 2023

• DOI för Thioacetalation and Multi-Component Thiomethylative Friedel-Crafts Arylation Using BF₃SMe₂
• Ladda ner fulltext (pdf) av Thioacetalation and Multi-Component Thiomethylative Friedel-Crafts Arylation Using BF₃SMe₂

On-Tissue Chemical Derivatization for Comprehensive Mapping of Brain Carboxyl and Aldehyde Metabolites by MALDI-MS Imaging

Kaya, Ibrahim; Schembri, Luke S; Nilsson, Anna; Shariatgorji, Reza et al.

Ingår i Journal of the American Society for Mass Spectrometry, s. 836-846, 2023

• DOI för On-Tissue Chemical Derivatization for Comprehensive Mapping of Brain Carboxyl and Aldehyde Metabolites by MALDI-MS Imaging
• Ladda ner fulltext (pdf) av On-Tissue Chemical Derivatization for Comprehensive Mapping of Brain Carboxyl and Aldehyde Metabolites by MALDI-MS Imaging

Acyl Amidines by Pd-Catalyzed Aminocarbonylation: One-Pot Cyclizations and C-11 Labeling

Rydfjord, Jonas; Roslin, Sara; Roy, Tamal; Abbas, Alaa et al.

Ingår i Journal of Organic Chemistry, s. 5078-5089, 2023

• DOI för Acyl Amidines by Pd-Catalyzed Aminocarbonylation: One-Pot Cyclizations and C-11 Labeling
• Ladda ner fulltext (pdf) av Acyl Amidines by Pd-Catalyzed Aminocarbonylation: One-Pot Cyclizations and C-11 Labeling

Prodrugs of the Archetypal Dynamin Inhibitor Bis-T-22

Odell, Luke R.; Robertson, Mark J.; Young, Kelly A.; McGeachie, Andrew B. et al.

Ingår i ChemMedChem, 2022

• DOI för Prodrugs of the Archetypal Dynamin Inhibitor Bis-T-22
• Ladda ner fulltext (pdf) av Prodrugs of the Archetypal Dynamin Inhibitor Bis-T-22

P-119 - Efficient cartridge-based synthesis of a novel [18F]tetrazine for large molecule labelling

Rokka, Johanna; Syvaenen, Stina; Odell, Luke R.; Schlein, Eva et al.

Ingår i Nuclear Medicine and Biology, 2022

• DOI för P-119 - Efficient cartridge-based synthesis of a novel [18F]tetrazine for large molecule labelling

Pyrimidyn‐Based Dynamin Inhibitors as Novel Cytotoxic Agents

Odell, Luke R.; Chau, Ngoc; Russell, Cecilia C.; Young, Kelly A. et al.

Ingår i ChemMedChem, 2022

• DOI för Pyrimidyn‐Based Dynamin Inhibitors as Novel Cytotoxic Agents

Region-Specific and Age-Dependent Multitarget Effects of Acetylcholinesterase Inhibitor Tacrine on Comprehensive Neurotransmitter Systems

Fridjonsdottir, Elva; Vallianatou, Theodosia; Mantas, Ioannis; Shariatgorji, Reza et al.

Ingår i ACS Chemical Biology, s. 147-158, 2022

• DOI för Region-Specific and Age-Dependent Multitarget Effects of Acetylcholinesterase Inhibitor Tacrine on Comprehensive Neurotransmitter Systems
• Ladda ner fulltext (pdf) av Region-Specific and Age-Dependent Multitarget Effects of Acetylcholinesterase Inhibitor Tacrine on Comprehensive Neurotransmitter Systems

Spatial visualization of comprehensive brain neurotransmitter systems and neuroactive substances by selective in situ chemical derivatization mass spectrometry imaging

Shariatgorji, Reza; Nilsson, Anna; Fridjonsdottir, Elva; Strittmatter, Nicole et al.

Ingår i Nature Protocols, s. 3298-3321, 2021

• DOI för Spatial visualization of comprehensive brain neurotransmitter systems and neuroactive substances by selective in situ chemical derivatization mass spectrometry imaging

Synthesis of substituted 3,4-dihydroquinazolinones via a metal free Leuckart-Wallach type reaction

Bokale-Shivale, Suvarna; Amin, Mohammad A.; Sawant, Rajiv T.; Stevens, Marc Y. et al.

Ingår i RSC Advances, s. 349-353, 2021

• DOI för Synthesis of substituted 3,4-dihydroquinazolinones via a metal free Leuckart-Wallach type reaction
• Ladda ner fulltext (pdf) av Synthesis of substituted 3,4-dihydroquinazolinones via a metal free Leuckart-Wallach type reaction

The Wittig Bioconjugation of Maleimide Derived, Water Soluble Phosphonium Ylides to Aldehyde-Tagged Proteins

Hartmann, Rafael W.; Pijnappel, Matthijs; Nilvebrant, Johan; Helgudottir, Hildur Run et al.

Ingår i Organic and biomolecular chemistry, s. 10417-10423, 2021

• DOI för The Wittig Bioconjugation of Maleimide Derived, Water Soluble Phosphonium Ylides to Aldehyde-Tagged Proteins
• Ladda ner fulltext (pdf) av The Wittig Bioconjugation of Maleimide Derived, Water Soluble Phosphonium Ylides to Aldehyde-Tagged Proteins

PET Imaging of GPR44 by Antagonist [C-11]MK-7246 in Pigs

Cheung, Pierre; Zhang, Bo; Puuvuori, Emmi; Estrada, Sergio et al.

Ingår i Biomedicines, 2021

• DOI för PET Imaging of GPR44 by Antagonist [C-11]MK-7246 in Pigs
• Ladda ner fulltext (pdf) av PET Imaging of GPR44 by Antagonist [C-11]MK-7246 in Pigs

Mass spectrometry imaging identifies abnormally elevated brain L-DOPA levels and extrastriatal monoaminergic dysregulation in L-DOPA-induced dyskinesia

Fridjonsdottir, Elva; Shariatgorji, Mohammadreza; Nilsson, Anna; Vallianatou, Theodosia et al.

Ingår i Science Advances, 2021

• DOI för Mass spectrometry imaging identifies abnormally elevated brain L-DOPA levels and extrastriatal monoaminergic dysregulation in L-DOPA-induced dyskinesia
• Ladda ner fulltext (pdf) av Mass spectrometry imaging identifies abnormally elevated brain L-DOPA levels and extrastriatal monoaminergic dysregulation in L-DOPA-induced dyskinesia

Sustainability in drug discovery

Wynendaele, Evelien; Furman, Christophe; Wielgomas, Bartosz; Larsson, Per et al.

Ingår i Medicine in Drug Discovery, 2021

• DOI för Sustainability in drug discovery
• Ladda ner fulltext (pdf) av Sustainability in drug discovery

Regio- and Stereoselective Synthesis of Allylic Spiroethers (Spirobenzofuranes) via an Intramolecular Mizoroki-Heck Reaction

Adeyemi, Ahmed; Odell, Luke R.; Larhed, Mats

Ingår i Journal of Organic Chemistry, s. 7648-7657, 2020

• DOI för Regio- and Stereoselective Synthesis of Allylic Spiroethers (Spirobenzofuranes) via an Intramolecular Mizoroki-Heck Reaction

Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.

Hartmann, Rafael; Fahrner, Raphael; Shevshenko, Denys; Fryknäs, Mårten et al.

Ingår i ChemMedChem, s. 2500-2512, 2020

• DOI för Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.
• Ladda ner fulltext (pdf) av Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.

Turning Information Dissipation into Dissemination: Instagram as a Communication Enhancing Tool during the COVID-19 Pandemic and Beyond

Ye, Sofie; Hartmann, Rafael; Söderström, Marcus; Amin, Mohammad A. et al.

Ingår i Journal of Chemical Education, s. 3217-3222, 2020

• DOI för Turning Information Dissipation into Dissemination: Instagram as a Communication Enhancing Tool during the COVID-19 Pandemic and Beyond

Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF₃⦁SMe₂

Söderström, Marcus; Zamaratski, Edouard; Odell, Luke R.

Ingår i European Journal of Organic Chemistry, s. 5402-5408, 2019

• DOI för Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF₃⦁SMe₂
• Ladda ner fulltext (pdf) av Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF₃⦁SMe₂

Synthesis and preclinical evaluation of the CRTH2 antagonist [¹¹C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

Eriksson, Jonas; Roy, Tamal; Sawadjoon, Supaporn; Bachmann, Kim et al.

Ingår i Nuclear Medicine and Biology, s. 1-10, 2019

• DOI för Synthesis and preclinical evaluation of the CRTH2 antagonist [¹¹C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass
• Ladda ner fulltext (pdf) av Synthesis and preclinical evaluation of the CRTH2 antagonist [¹¹C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

Comprehensive mapping of neurotransmitter networks by MALDI-MS imaging

Shariatgorji, Mohammadreza; Nilsson, Anna; Fridjonsdottir, Elva; Vallianatou, Theodosia et al.

Ingår i Nature Methods, s. 1021-1028, 2019

• DOI för Comprehensive mapping of neurotransmitter networks by MALDI-MS imaging

Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

Schembri, Luke S; Eriksson, Jonas; Odell, Luke R.

Ingår i Journal of Organic Chemistry, s. 6970-6981, 2019

• DOI för Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

Palladium-Catalyzed Molybdenum Hexacarbonyl-Mediated Gas-Free Carbonylative Reactions

Åkerbladh, Linda; Odell, Luke R.; Larhed, Mats

Ingår i Synlett, s. 141-155, 2019

• DOI för Palladium-Catalyzed Molybdenum Hexacarbonyl-Mediated Gas-Free Carbonylative Reactions

Microwave-Assisted aza-Friedel-Crafts Arylation of N-Acyliminium Ions: Expedient Access to 4 -Aryl 3,4-Dihydroquinazolinones

Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

Ingår i ACS Omega, s. 14258-14265, 2018

• DOI för Microwave-Assisted aza-Friedel-Crafts Arylation of N-Acyliminium Ions: Expedient Access to 4 -Aryl 3,4-Dihydroquinazolinones
• Ladda ner fulltext (pdf) av Microwave-Assisted aza-Friedel-Crafts Arylation of N-Acyliminium Ions: Expedient Access to 4 -Aryl 3,4-Dihydroquinazolinones

Carbonylations beyond aryl-X: Development of new multicomponent reactions

Odell, Luke R.; Åkerbladh, Linda; Schembri, Luke S; Nordeman, Patrik et al.

Ingår i Abstracts of Papers of the American Chemical Society, 2018

Synthesis of ¹¹C-Labelled Ureas by Palladium(II)-Mediated Oxidative Carbonylation

Bergman, Sara; Brandt, Peter; Nordeman, Patrik; Larhed, Mats et al.

Ingår i Molecules, 2017

• DOI för Synthesis of ¹¹C-Labelled Ureas by Palladium(II)-Mediated Oxidative Carbonylation
• Ladda ner fulltext (pdf) av Synthesis of ¹¹C-Labelled Ureas by Palladium(II)-Mediated Oxidative Carbonylation

Palladium-mediated C-11-carbonylations using aryl halides and cyanamide

Nordeman, Patrik; Chow, Shiao Y.; Odell, A. F.; Antoni, Gunnar et al.

Ingår i Organic and biomolecular chemistry, s. 4875-4881, 2017

• DOI för Palladium-mediated C-11-carbonylations using aryl halides and cyanamide

Synthesis of N-Sulfonyl Amidines and Acyl Sulfonyl Ureas from Sulfonyl Azides, Carbon Monoxide, and Amides

Chow, Shiao Y.; Odell, Luke R.

Ingår i Journal of Organic Chemistry, s. 2515-2522, 2017

• DOI för Synthesis of N-Sulfonyl Amidines and Acyl Sulfonyl Ureas from Sulfonyl Azides, Carbon Monoxide, and Amides

Acetic acid-promoted cascade N-acyliminium ion/aza-Prins cyclization: stereoselective synthesis of functionalized fused tricyclic piperidines

Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

Ingår i Chemical Communications, s. 2110-2113, 2017

• DOI för Acetic acid-promoted cascade N-acyliminium ion/aza-Prins cyclization: stereoselective synthesis of functionalized fused tricyclic piperidines

Low-Pressure Radical 11C-Aminocarbonylation of Alkyl Iodides through Thermal Initiation

Chow, Shiao Y.; Odell, Luke R.; Eriksson, Jonas

Ingår i European Journal of Organic Chemistry, s. 1236-1236, 2017

• DOI för Low-Pressure Radical 11C-Aminocarbonylation of Alkyl Iodides through Thermal Initiation

Synthesis of 4H-Benzo[e][1,3]oxazin-4-ones by a Carbonylation-Cyclization Domino Reaction of ortho-Halophenols and Cyanamide

Åkerbladh, Linda; Chow, Shiao Y.; Odell, Luke R.; Larhed, Mats

Ingår i ChemistryOpen, s. 620-628, 2017

• DOI för Synthesis of 4H-Benzo[e][1,3]oxazin-4-ones by a Carbonylation-Cyclization Domino Reaction of ortho-Halophenols and Cyanamide
• Ladda ner fulltext (pdf) av Synthesis of 4H-Benzo[e][1,3]oxazin-4-ones by a Carbonylation-Cyclization Domino Reaction of ortho-Halophenols and Cyanamide

Palladium and Visible-Light Mediated Carbonylative Suzuki-Miyaura Coupling of Unactivated Alkyl Halides and Aryl Boronic Acids

Roslin, Sara; Odell, Luke R.

Ingår i Chemical Communications, s. 6895-6898, 2017

• DOI för Palladium and Visible-Light Mediated Carbonylative Suzuki-Miyaura Coupling of Unactivated Alkyl Halides and Aryl Boronic Acids

Synthesis and In Vitro Evaluation of 5-Substituted Benzovesamicol Analogs containing N-Substituted Amides as Potential Positron Emission Tomography Tracers for the Vesicular Acetylcholine Transporter

Roslin, Sara; De Rosa, Maria; Deuther-Conrad, Winnie; Eriksson, Jonas et al.

Ingår i Bioorganic & Medicinal Chemistry, s. 5095-5106, 2017

• DOI för Synthesis and In Vitro Evaluation of 5-Substituted Benzovesamicol Analogs containing N-Substituted Amides as Potential Positron Emission Tomography Tracers for the Vesicular Acetylcholine Transporter

Palladium(0)-Catalyzed Carbonylative One-Pot Synthesis of N-Acylguanidines

Åkerbladh, Linda; Schembri, Luke S; Larhed, Mats; Odell, Luke R.

Ingår i Journal of Organic Chemistry, s. 12520-12529, 2017

• DOI för Palladium(0)-Catalyzed Carbonylative One-Pot Synthesis of N-Acylguanidines

Route to 3-Amidino Indoles via Pd(II)-Catalyzed C-H Bond Activation

Rydfjord, Jonas; Skillinghaug, Bobo; Brandt, Peter; Odell, Luke R. et al.

Ingår i Organic Letters, s. 4066-4069, 2017

• DOI för Route to 3-Amidino Indoles via Pd(II)-Catalyzed C-H Bond Activation

Pyrimidine-Based Inhibitors of Dynamin I GTPase Activity: Competitive Inhibition at the Pleckstrin Homology Domain

Odell, Luke R.; Abdel-Hamid, Mohammed K.; Hill, Timothy A.; Chau, Ngoc et al.

Ingår i Journal of Medicinal Chemistry, s. 349-361, 2017

• DOI för Pyrimidine-Based Inhibitors of Dynamin I GTPase Activity: Competitive Inhibition at the Pleckstrin Homology Domain

Synthesis of C-11-labeled Sulfonyl Carbamates through a Multicomponent Reaction Employing Sulfonyl Azides, Alcohols, and [C-11]CO

Stevens, Marc; Chow, Shiao; Estrada, Sergio; Eriksson, Jonas et al.

Ingår i ChemistryOpen, s. 566-573, 2016

• DOI för Synthesis of C-11-labeled Sulfonyl Carbamates through a Multicomponent Reaction Employing Sulfonyl Azides, Alcohols, and [C-11]CO
• Ladda ner fulltext (pdf) av Synthesis of C-11-labeled Sulfonyl Carbamates through a Multicomponent Reaction Employing Sulfonyl Azides, Alcohols, and [C-11]CO

Low-Pressure Radical C-11-Aminocarbonylation of Alkyl Iodides through Thermal Initiation

Chow, Shiao Y.; Odell, Luke R.; Eriksson, Jonas

Ingår i European Journal of Organic Chemistry, s. 5980-5989, 2016

• DOI för Low-Pressure Radical C-11-Aminocarbonylation of Alkyl Iodides through Thermal Initiation

Synthesis of ¹¹C-labelled Sulfonyl Carbamates via a Multicomponent Reaction Employing Sulfonyl Azides, Alcohols and [¹¹C]CO

Stevens, Marc; Chow, Chow; Estrada, Sergio; Eriksson, Jonas et al.

Ingår i ChemistryOpen, s. 566-573, 2016

• DOI för Synthesis of ¹¹C-labelled Sulfonyl Carbamates via a Multicomponent Reaction Employing Sulfonyl Azides, Alcohols and [¹¹C]CO
• Ladda ner fulltext (pdf) av Synthesis of ¹¹C-labelled Sulfonyl Carbamates via a Multicomponent Reaction Employing Sulfonyl Azides, Alcohols and [¹¹C]CO

Mild and Low-Pressure fac-Ir(ppy)3-Mediated Radical Aminocarbonylation of Unactivated Alkyl Iodides through Visible-Light Photoredox Catalysis

Chow, Shiao Y.; Stevens, Marc; Åkerbladh, Linda; Bergman, Sara et al.

Ingår i Chemistry - A European Journal, s. 9155-9161, 2016

• DOI för Mild and Low-Pressure fac-Ir(ppy)3-Mediated Radical Aminocarbonylation of Unactivated Alkyl Iodides through Visible-Light Photoredox Catalysis

Microwave-Assisted Branching Cascades: A Route to Diverse 3,4-Dihydroquinazolinone-Embedded Polyheterocyclic Scaffolds

Sawant, Rajiv T.; Stevens, Marc Y.; Sköld, Christian; Odell, Luke R.

Ingår i Organic Letters, s. 5392-5395, 2016

• DOI för Microwave-Assisted Branching Cascades: A Route to Diverse 3,4-Dihydroquinazolinone-Embedded Polyheterocyclic Scaffolds

Synthesis of sodium aryl sulfinates from aryl bromides employing 1,4-diazabicyclo[2.2.2]octane bis(sulfur dioxide) adduct (DABSO) as a bench-stable, gas-free alternative to SO2

Skillinghaug, Bobo; Rydfjord, Jonas; Odell, Luke R.

Ingår i Tetrahedron Letters, s. 533-536, 2016

• DOI för Synthesis of sodium aryl sulfinates from aryl bromides employing 1,4-diazabicyclo[2.2.2]octane bis(sulfur dioxide) adduct (DABSO) as a bench-stable, gas-free alternative to SO2

Sulfonyl Azides as Precursors in Ligand-free Palladium-Catalyzed Synthesis of Sulfonyl Carbamates and Sulfonyl Ureas and Synthesis of Sulfonamides

Chow, Shiao; Stevens, Marc; Odell, Luke

Ingår i Journal of Organic Chemistry, s. 2681-2691, 2016

• DOI för Sulfonyl Azides as Precursors in Ligand-free Palladium-Catalyzed Synthesis of Sulfonyl Carbamates and Sulfonyl Ureas and Synthesis of Sulfonamides

Synthesis of 2-Aminoquinazolinones via Carbonylative Coupling of ortho-lodoanilines and Cyanamide

Åkerbladh, Linda; Odell, Luke R.

Ingår i Journal of Organic Chemistry, s. 2966-2973, 2016

• DOI för Synthesis of 2-Aminoquinazolinones via Carbonylative Coupling of ortho-lodoanilines and Cyanamide

A microwave-assisted multicomponent synthesis of substituted 3,4-dihydroquinazolinones

Stevens, Marc; Wieckowski, Krzysztof; Wu, Peng; Sawant, Rajiv T et al.

Ingår i Organic and biomolecular chemistry, s. 2044-2054, 2015

• DOI för A microwave-assisted multicomponent synthesis of substituted 3,4-dihydroquinazolinones

3,4-Dihydro-3-(2-hydroxyethyl)-4-(nitromethyl)quinazolin-2(1H)-one

Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

Ingår i Molbank, 2015

• DOI för 3,4-Dihydro-3-(2-hydroxyethyl)-4-(nitromethyl)quinazolin-2(1H)-one
• Ladda ner fulltext (pdf) av 3,4-Dihydro-3-(2-hydroxyethyl)-4-(nitromethyl)quinazolin-2(1H)-one

Synthesis of 4-Quinolones via a Carbonylative Sonogashira Cross-Coupling Using Molybdenum Hexacarbonyl as a CO Source

Åkerbladh, Linda; Nordeman, Patrik; Wejdemar, Matyas; Odell, Luke R. et al.

Ingår i Journal of Organic Chemistry, s. 1464-1471, 2015

• DOI för Synthesis of 4-Quinolones via a Carbonylative Sonogashira Cross-Coupling Using Molybdenum Hexacarbonyl as a CO Source

Cyclic amidines as precursors for imidazoles

Stevens, Marc Y.; Rozycka-Sokolowska, Ewa; Andersson, Gabriella; Odell, Luke R. et al.

Ingår i ARKIVOC, s. 219-229, 2015

• DOI för Cyclic amidines as precursors for imidazoles
• Ladda ner fulltext (pdf) av Cyclic amidines as precursors for imidazoles

Rapid Access to Polyfunctionalized 3,4-Dihydroquinazolinones through a Sequential N-Acyliminium Ion Mannich Reaction Cascade

Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

Ingår i European Journal of Organic Chemistry, s. 7743-7755, 2015

• DOI för Rapid Access to Polyfunctionalized 3,4-Dihydroquinazolinones through a Sequential N-Acyliminium Ion Mannich Reaction Cascade

1,8-Naphthalimide derivatives: new leads against dynamin I GTPase activity.

Abdel-Hamid, Mohammed K; Macgregor, Kylie A; Odell, Luke R; Chau, Ngoc et al.

Ingår i Organic and biomolecular chemistry, 2015

• DOI för 1,8-Naphthalimide derivatives: new leads against dynamin I GTPase activity.

Synthesis of arylsulfonyl azides via diazotransfer using an imidazole-1-sulfonyl azide salt: Scope and N-15 NMR labeling experiments

Stevens, Marc Y.; Sawant, Rajiv T.; Odell, Luke R.

Ingår i Abstracts of Papers of the American Chemical Society, 2014

Synthesis and evaluation of isoleucine derived angiotensin II AT(2) receptor ligands

Veron, Jean-Baptiste; Joshi, Advait; Wallinder, Charlotta; Larhed, Mats et al.

Ingår i Bioorganic & Medicinal Chemistry Letters, s. 476-479, 2014

• DOI för Synthesis and evaluation of isoleucine derived angiotensin II AT(2) receptor ligands

Development of quinone analogues as dynamin GTPase inhibitors

MacGregor, Kylie A; Abdel-Hamid, Mohammed K; Odell, Luke R; Chau, Ngoc et al.

Ingår i European Journal of Medicinal Chemistry, s. 191-206, 2014

• DOI för Development of quinone analogues as dynamin GTPase inhibitors

11C-Labeling of a Potent Hydroxyethylamine BACE-1 Inhibitor and Evaluation in vitro and in vivo

Nordeman, Patrik; Estrada, Sergio; Odell, Luke R; Larhed, Mats et al.

Ingår i Nuclear Medicine and Biology, s. 536-543, 2014

• DOI för 11C-Labeling of a Potent Hydroxyethylamine BACE-1 Inhibitor and Evaluation in vitro and in vivo

C-11-Labeling of a potent hydroxyethylamine BACE-1 inhibitor and evaluation in vitro and in vivo

Nordeman, Patrik; Estrada, Sergio; Odell, Luke; Larhed, Mats et al.

Ingår i Nuclear Medicine and Biology, s. 536-543, 2014

• DOI för C-11-Labeling of a potent hydroxyethylamine BACE-1 inhibitor and evaluation in vitro and in vivo

An Improved Palladium(II)-Catalyzed Method for the Synthesis of Aryl Ketones from Aryl Carboxylic Acids and Organonitriles

Axelsson, Linda; Veron, Jean-Baptiste; Sävmarker, Jonas; Lindh, Jonas et al.

Ingår i Tetrahedron Letters, s. 2376-2380, 2014

• DOI för An Improved Palladium(II)-Catalyzed Method for the Synthesis of Aryl Ketones from Aryl Carboxylic Acids and Organonitriles

Synthesis of sulfonyl azides via diazotransfer using an imidazole-1-sulfonyl azide salt: scope and ¹⁵N NMR labeling experiments

Stevens, Marc; Sawant, Rajiv; Odell, Luke

Ingår i Journal of Organic Chemistry, s. 4826-4831, 2014

• DOI för Synthesis of sulfonyl azides via diazotransfer using an imidazole-1-sulfonyl azide salt: scope and ¹⁵N NMR labeling experiments

Palladium-Catalyzed Carbonylative Synthesis of N-Cyanobenzamides from Aryl Iodides/Bromides and Cyanamide

Mane, Rajendra S; Nordeman, Patrik; Odell, Luke R; Larhed, Mats

Ingår i Tetrahedron Letters, s. 6912-6915, 2013

• DOI för Palladium-Catalyzed Carbonylative Synthesis of N-Cyanobenzamides from Aryl Iodides/Bromides and Cyanamide

Decarboxylative Palladium(II)-Catalyzed Synthesis of Aryl Amidines from Aryl Carboxylic Acids: Development and Mechanistic Investigation

Rydfjord, Jonas; Svensson, Fredrik; Trejos, Alejandro; Sjöberg, Per J. R. et al.

Ingår i Chemistry - A European Journal, s. 13803-13810, 2013

• DOI för Decarboxylative Palladium(II)-Catalyzed Synthesis of Aryl Amidines from Aryl Carboxylic Acids: Development and Mechanistic Investigation

Pyrimidyn Compounds: Dual-Action Small Molecule Pyrimidine-Based Dynamin Inhibitors

McGeachie, Andrew B; Odell, Luke R; Quan, Annie; Daniel, James A et al.

Ingår i ACS Chemical Biology, s. 1507-1518, 2013

• DOI för Pyrimidyn Compounds: Dual-Action Small Molecule Pyrimidine-Based Dynamin Inhibitors

A Novel p53 Mutant Found in Iatrogenic Urothelial Cancers Is Dysfunctional and Can Be Rescued by a Second-site Global Suppressor Mutation

Odell, Adam F; Odell, Luke R; Askham, Jon M; Alogheli, Hiba et al.

Ingår i Journal of Biological Chemistry, s. 16704-16714, 2013

• DOI för A Novel p53 Mutant Found in Iatrogenic Urothelial Cancers Is Dysfunctional and Can Be Rescued by a Second-site Global Suppressor Mutation

Organocatalytic asymmetric cross-aldol reaction of 2-chloroethoxy acetaldehyde: diversity-oriented synthesis of chiral substituted 1,4-dioxanes and morpholines

Sawant, Rajiv T.; Stevenson, Joanne; Odell, Luke R.; Arvidsson, Per I.

Ingår i Tetrahedron, s. 134-141, 2013

• DOI för Organocatalytic asymmetric cross-aldol reaction of 2-chloroethoxy acetaldehyde: diversity-oriented synthesis of chiral substituted 1,4-dioxanes and morpholines

Synthesis, biological evaluation and X-ray crystallographic studies of imidazo[1,2-a]-pyridine based Mycobacterium tuberculosis glutamine synthetase inhibitors

Nordqvist, Anneli; Nilsson, Mikael T.; Lagerlund, Olof; Muthas, Daniel et al.

Ingår i MedChemComm, s. 620-626, 2012

• DOI för Synthesis, biological evaluation and X-ray crystallographic studies of imidazo[1,2-a]-pyridine based Mycobacterium tuberculosis glutamine synthetase inhibitors

Molybdenum Hexacarbonyl Mediated CO Gas-Free Carbonylative Reactions

Odell, Luke R.; Russo, Francesco; Larhed, Mats

Ingår i Synlett, s. 685-698, 2012

• DOI för Molybdenum Hexacarbonyl Mediated CO Gas-Free Carbonylative Reactions

Aminocarbonylations Employing Mo(CO)(6) and a Bridged Two-Vial System: Allowing the Use of Nitro Group Substituted Aryl Iodides and Aryl Bromides

Nordeman, Patrik; Odell, Luke R; Larhed, Mats

Ingår i Journal of Organic Chemistry, s. 11393-11398, 2012

• DOI för Aminocarbonylations Employing Mo(CO)(6) and a Bridged Two-Vial System: Allowing the Use of Nitro Group Substituted Aryl Iodides and Aryl Bromides

Direct Palladium(II)-Catalyzed Synthesis of Arylamidines from Aryltrifluoroborates

Sävmarker, Jonas; Rydfjord, Jonas; Gising, Johan; Odell, Luke R. et al.

Ingår i Organic Letters, s. 2394-2397, 2012

• DOI för Direct Palladium(II)-Catalyzed Synthesis of Arylamidines from Aryltrifluoroborates

Trisubstituted Imidazoles as Mycobacterium tuberculosis Glutamine Synthetase Inhibitors

Gising, Johan; Nilsson, Mikael T; Odell, Luke R; Yahiaoui, Samir et al.

Ingår i Journal of Medicinal Chemistry, s. 2894-2898, 2012

• DOI för Trisubstituted Imidazoles as Mycobacterium tuberculosis Glutamine Synthetase Inhibitors
• Ladda ner fulltext (pdf) av Trisubstituted Imidazoles as Mycobacterium tuberculosis Glutamine Synthetase Inhibitors

Development of Stereocontrolled Palladium(II)-Catalyzed Domino Heck/Suzuki β, α-Diarylation Reactions with Chelating Vinyl Ethers and Arylboronic Acids

Trejos, Alejandro; Odell, Luke R.; Larhed, Mats

Ingår i ChemistryOpen, s. 49-56, 2012

• DOI för Development of Stereocontrolled Palladium(II)-Catalyzed Domino Heck/Suzuki β, α-Diarylation Reactions with Chelating Vinyl Ethers and Arylboronic Acids
• Ladda ner fulltext (pdf) av Development of Stereocontrolled Palladium(II)-Catalyzed Domino Heck/Suzuki β, α-Diarylation Reactions with Chelating Vinyl Ethers and Arylboronic Acids

Transmetallation Versus β-Hydride Elimination: The Role of 1,4 Benzoquinone in Chelation-Controlled Arylation Reactions with Arylboronic Acids

Sköld, Christian; Kleimark, Jonatan; Trejos, Alejandro; Odell, Luke R. et al.

Ingår i Chemistry - A European Journal, s. 4714-4722, 2012

• DOI för Transmetallation Versus β-Hydride Elimination: The Role of 1,4 Benzoquinone in Chelation-Controlled Arylation Reactions with Arylboronic Acids
• Ladda ner fulltext (pdf) av Transmetallation Versus β-Hydride Elimination: The Role of 1,4 Benzoquinone in Chelation-Controlled Arylation Reactions with Arylboronic Acids

Microwave-assisted synthesis of small molecules targeting the infectious diseases tuberculosis, HIV/AIDS, malaria and hepatitis C

Gising, Johan; Odell, Luke R.; Larhed, Mats

Ingår i Organic and biomolecular chemistry, s. 2713-2729, 2012

• DOI för Microwave-assisted synthesis of small molecules targeting the infectious diseases tuberculosis, HIV/AIDS, malaria and hepatitis C

Richard F. Heck: Nobel Laureate in Chemistry

Odell, Luke R; Larhed, Mats

Ingår i Les Prix Nobel, s. 133-138, 2011

A microwave-assisted, propylphosphonic anhydride (T3P (R)) mediated one-pot Fischer indole synthesis

Desroses, Matthieu; Wieckowski, Krzysztof; Stevens, Marc; Odell, Luke R.

Ingår i Tetrahedron Letters, s. 4417-4420, 2011

• DOI för A microwave-assisted, propylphosphonic anhydride (T3P (R)) mediated one-pot Fischer indole synthesis

Microwave-Assisted Synthesis of Weinreb and MAP Aryl Amides via Pd-Catalyzed Heck Aminocarbonylation Using Mo(CO)(6) or W(CO)(6)

Wieckowska, Anna; Fransson, Rebecca; Odell, Luke R.; Larhed, Mats

Ingår i Journal of Organic Chemistry, s. 978-981, 2011

• DOI för Microwave-Assisted Synthesis of Weinreb and MAP Aryl Amides via Pd-Catalyzed Heck Aminocarbonylation Using Mo(CO)(6) or W(CO)(6)

Iminochromene Inhibitors of Dynamins I and II GTPase Activity and Endocytosis

Hill, Timothy A.; Mariana, Anna; Gordon, Christopher P.; Odell, Luke R. et al.

Ingår i Journal of Medicinal Chemistry, s. 4094-4102, 2010

• DOI för Iminochromene Inhibitors of Dynamins I and II GTPase Activity and Endocytosis

The Pthaladyns: GTP Competitive Inhibitors of Dynamin I and II GTPase Derived from Virtual Screening

Odell, Luke R; Howan, Dian; Gordon, Christopher P.; Robertson, Mark J. et al.

Ingår i Journal of Medicinal Chemistry, s. 5267-5280, 2010

• DOI för The Pthaladyns: GTP Competitive Inhibitors of Dynamin I and II GTPase Derived from Virtual Screening

Continuous Flow Palladium(II): Catalyzed Oxidative Heck Reactions with Arylboronic Acids

Odell, Luke R.; Lindh, Jonas; Gustafsson, Tomas; Larhed, Mats

Ingår i European Journal of Organic Chemistry, s. 2270-2274, 2010

• DOI för Continuous Flow Palladium(II): Catalyzed Oxidative Heck Reactions with Arylboronic Acids

Functionalized 3-amino-imidazo[1,2-a]pyridines: A novel class of drug-like Mycobacterium tuberculosis glutamine synthetase inhibitors

Odell, Luke R.; Nilsson, Mikael T.; Gising, Johan; Lagerlund, Olof et al.

Ingår i Bioorganic & Medicinal Chemistry Letters, s. 4790-4793, 2009

• DOI för Functionalized 3-amino-imidazo[1,2-a]pyridines: A novel class of drug-like Mycobacterium tuberculosis glutamine synthetase inhibitors

Azido and diazarinyl analogues of bis-tyrphostin as asymmetrical inhibitors of dynamin GTPase

Odell, Luke R; Chau, Ngoc; Mariana, Anna; Graham, Mark E et al.

Ingår i ChemMedChem, s. 1182-1188, 2009

• DOI för Azido and diazarinyl analogues of bis-tyrphostin as asymmetrical inhibitors of dynamin GTPase

Inhibition of dynamin mediated endocytosis by the dynoles: synthesis and functional activity of a family of indoles

Hill, Timothy A; Gordon, Christopher P; McGeachie, Andrew B; Venn-Brown, Barbara et al.

Ingår i Journal of Medicinal Chemistry, s. 3762-3773, 2009

• DOI för Inhibition of dynamin mediated endocytosis by the dynoles: synthesis and functional activity of a family of indoles

A versatile new synthetic route to 1N-hydroxyindazoles

Lehmann, Fredrik; Koolmeister, Tobias; Odell, Luke R; Scobie, Martin

Ingår i Organic Letters, s. 5078-5081, 2009

• DOI för A versatile new synthetic route to 1N-hydroxyindazoles

Microwave-promoted aminocarbonylation of aryl triflates using Mo(CO)₆ as a solid CO source

Odell, Luke R.; Sävmarker, Jonas; Larhed, Mats

Ingår i Tetrahedron Letters, s. 6115-6118, 2008

• DOI för Microwave-promoted aminocarbonylation of aryl triflates using Mo(CO)₆ as a solid CO source

Evaluation of the amino acid binding site of Mycobacterium tuberculosis glutamine synthetase for drug discovery

Nordqvist, Anneli; Nilsson, Mikael T.; Röttger, Svenja; Odell, Luke R. et al.

Ingår i Bioorganic & Medicinal Chemistry, s. 5501-5513, 2008

• DOI för Evaluation of the amino acid binding site of Mycobacterium tuberculosis glutamine synthetase for drug discovery
• Ladda ner fulltext (pdf) av Evaluation of the amino acid binding site of Mycobacterium tuberculosis glutamine synthetase for drug discovery

Isolation and identification of unique marker compounds from the Tasmanian poppy Papaver somniferum N. Implications for the identification of illicit heroin of Tasmanian origin.

Odell, Luke R; Skopec, Jana; McCluskey, Adam

Ingår i Forensic Science International, 2008

• DOI för Isolation and identification of unique marker compounds from the Tasmanian poppy Papaver somniferum N. Implications for the identification of illicit heroin of Tasmanian origin.

Microwave-enhanced alpha-arylation of a protected glycine in water: evaluation of 3-phenylglycine derivatives as inhibitors of the tuberculosis enzyme, glutamine synthetase

Lagerlund, Olof; Odell, Luke R.; Mowbray, Sherry L.; Nilsson, Mikael T. et al.

Ingår i Combinatorial chemistry & high throughput screening, s. 783-789, 2007

• DOI för Microwave-enhanced alpha-arylation of a protected glycine in water: evaluation of 3-phenylglycine derivatives as inhibitors of the tuberculosis enzyme, glutamine synthetase

Crystal and Molecular Structures of Benzyl-(2-chloro-6-methylpyrimidin-4-yl)amine and Benzyl-(4-chloro-6-methylpyrimidin-2-yl)amine: Confirmation of Computationally Predicted Restricted Rotation

Odell, Luke R.; McCluskey, Adam; Failes, Timothy W.; Tiekink, Edward R. T.

Ingår i Journal of Chemical Crystallography, s. 817-824, 2007

• DOI för Crystal and Molecular Structures of Benzyl-(2-chloro-6-methylpyrimidin-4-yl)amine and Benzyl-(4-chloro-6-methylpyrimidin-2-yl)amine: Confirmation of Computationally Predicted Restricted Rotation

A 'cold synthesis' of heroin and implications in heroin signature analysis utility of trifluoroacetic/acetic anhydride in the acetylation of morphine.

Odell, Luke R; Skopec, Jana; McCluskey, Adam

Ingår i Forensic Science International, 2006

• DOI för A 'cold synthesis' of heroin and implications in heroin signature analysis utility of trifluoroacetic/acetic anhydride in the acetylation of morphine.

BiCl3-mediated opening of epoxides, a facile route to chlorohydrins or amino alcohols: one reagent, two paths

McCluskey, Adam; Leitch, Sarah K.; Garner, James; Caden, Christine E. et al.

Ingår i Tetrahedron Letters, s. 8229-8232, 2005

• DOI för BiCl3-mediated opening of epoxides, a facile route to chlorohydrins or amino alcohols: one reagent, two paths

Small molecule inhibitors of dynamin I GTPase activity: development of dimeric tyrphostins.

Hill, Timothy; Odell, Luke R; Edwards, Jennifer K; Graham, Mark E et al.

Ingår i Journal of Medicinal Chemistry, 2005

• DOI för Small molecule inhibitors of dynamin I GTPase activity: development of dimeric tyrphostins.

Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity.

Hill, Timothy A; Odell, Luke R; Quan, Annie; Abagyan, Ruben et al.

Ingår i Bioorganic & Medicinal Chemistry Letters, 2004

• DOI för Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity.

Identification of Aminopyrimidine Regioisomers via Line Broadening Effects in 1H and 13C NMR Spectroscopy

Garner, J.; Hill, T.; Odell, L.R.; Keller, P. et al.

Ingår i Australian Journal of Chemistry, s. 1079-1083, 2004

Visible-Light Photocatalysis as an Enabling Tool for the Functionalization of Unactivated C(sp(3))-Substrates

Roslin, Sara; Odell, Luke R.

Ingår i European Journal of Organic Chemistry, s. 1993-2007, 2017

• DOI för Visible-Light Photocatalysis as an Enabling Tool for the Functionalization of Unactivated C(sp(3))-Substrates

Inhibition of Glutamine Synthetase: A Potential Drug Target in Mycobacterium tuberculosis

Mowbray, Sherry L; Kathiravan, Muthu K; Pandey, Abhishek A; Odell, Luke R

Ingår i Molecules, s. 13161-13176, 2014

• DOI för Inhibition of Glutamine Synthetase: A Potential Drug Target in Mycobacterium tuberculosis
• Ladda ner fulltext (pdf) av Inhibition of Glutamine Synthetase: A Potential Drug Target in Mycobacterium tuberculosis

Aspartic protease inhibitors containing tertiary alcohol transition-state mimics

Motwani, Hitesh V.; De Rosa, Maria; Odell, Luke R.; Hallberg, Anders et al.

Ingår i European Journal of Medicinal Chemistry, s. 462-490, 2014

• DOI för Aspartic protease inhibitors containing tertiary alcohol transition-state mimics

Syntheses of new tuberculosis inhibitors promoted by microwave irradiation

De Rosa, Maria; Gising, Johan; Odell, Luke R; Larhed, Mats

Ingår i Upsala Journal of Medical Sciences, s. 181-191, 2014

• DOI för Syntheses of new tuberculosis inhibitors promoted by microwave irradiation

Microwave-assisted synthesis of anti-tuberculosis, HIV and hepatitis C agents

Gising, Johan; Larhed, Mats; Odell, Luke R

Ingår i Microwaves in Drug Discovery and Development, s. 34-54, Future Medicine, 2014

• DOI för Microwave-assisted synthesis of anti-tuberculosis, HIV and hepatitis C agents

7.18 Addition Reactions with Formation of Carbon–Carbon Bonds: (v) The Oxidative Heck Reaction

Odell, L. R.; Sävmarker, J.; Lindh, J.; Nilsson, P. et al.

Ingår i Comprehensive Organic Synthesis II (Second Edition), s. 492-537, Elsevier, 2014

Alkenes with Metal-Directing Groups as Reaction Components

Trejos, Alejandro; Odell, Luke R

Ingår i Science of Synthesis: Cross-Coupling and Heck-Type Reactions, Volume 3, Metal-Catalyzed Heck-Type Reactions and C-C Cross Coupling via C–H Activation, s. 345-390, Georg Thieme Verlag KG, 2013

Microwave-Heated Transition Metal-Catalyzed Coupling Reactions

Russo, Francesco; Odell, Luke R; Olofsson, Kristofer; Nilsson, Peter et al.

Ingår i Microwaves in Organic Synthesis, s. 607-672, Wiley-VCH Verlagsgesellschaft, 2012

Microwave-Assisted Transition Metal-Catalyzed Asymmetric Synthesis

Odell, Luke R; Larhed, Mats

Ingår i Catalytic Methods in Asymmetric Synthesis, s. 391-412, Wiley-Blackwell, 2011

• DOI för Microwave-Assisted Transition Metal-Catalyzed Asymmetric Synthesis

Microwave-accelerated homogenous catalysis in water

Odell, Luke R; Larhed, Mats

Ingår i Handbook of green chemistry, s. 79-99, Wiley-VCH Verlagsgesellschaft, 2009

Late-Stage Defluorinative Functionalization: Synthesis of Methyl-Dithioesters and Thioamides from Trifluoromethylarenes

Söderström, Marcus; Odell, Luke R.