Publications

A novel ¹⁸F-labelled tetrazine ester prosthetic group for improved radiolabelling and in vivo stability of proteins and peptides

Lechi, Francesco; Odell, Luke R.; Wegrzyniak, Olivia; Balestri, Lorenzo et al.

Part of EJNMMI Radiopharmacy and Chemistry, 2026

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• DOI for A novel ¹⁸F-labelled tetrazine ester prosthetic group for improved radiolabelling and in vivo stability of proteins and peptides
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Ascending single-dose study of the safety, pharmacokinetics, and pharmacodynamics of CSTI-500, a novel monoamine triple reuptake inhibitor, first-in-human

Appel, Lieuwe; Risinger, Robert; Wall, Anders; Murck, Harald et al.

Part of Psychopharmacology, p. 565-580, 2026

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• DOI for Ascending single-dose study of the safety, pharmacokinetics, and pharmacodynamics of CSTI-500, a novel monoamine triple reuptake inhibitor, first-in-human
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From virtual screening to selective angiotensin II type 2 receptor ligands: discovery of a novel scaffold

Patel, Jayendra Z.; Sandberg, Lars; Wannberg, Johan; Söderström, Marcus et al.

Part of Results in Chemistry, 2026

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• DOI for From virtual screening to selective angiotensin II type 2 receptor ligands: discovery of a novel scaffold
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Heterocyclic scaffold-fused dimethoxy-dibenzocyclooctynes for photoactivatable click chemistry

Larsson, N. Alfred; Jo, Taegeun; Bremberg, Ulf; Crespi, Stefano et al.

Part of Organic and biomolecular chemistry, p. 120-126, 2026

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• DOI for Heterocyclic scaffold-fused dimethoxy-dibenzocyclooctynes for photoactivatable click chemistry
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Late-stage defluorinative functionalization: synthesis of thio-amides and heterocycles from trifluoromethylarenes

Söderström, Marcus; Olaniran Håkansson, Esther; Odell, Luke R.

Part of Organic Chemistry Frontiers, p. 1275-1280, 2026

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• DOI for Late-stage defluorinative functionalization: synthesis of thio-amides and heterocycles from trifluoromethylarenes
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Low-dose testosterone administration and oestrogen synthase availability in the female brain: A pilot study

Dubol, Manon; Jonasson, My; Takahashi, Kayo; Wikström, Johan et al.

Part of Journal of neuroendocrinology, 2026

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• DOI for Low-dose testosterone administration and oestrogen synthase availability in the female brain: A pilot study
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New high affinity AT2 receptor ligands comprising a 2-methyl substituted phenylthiophene scaffold

Gising, Johan; Wannberg, Johan; Isaksson, Rebecka; Sallander, Jessica et al.

Part of Bioorganic & Medicinal Chemistry, 2026

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• DOI for New high affinity AT2 receptor ligands comprising a 2-methyl substituted phenylthiophene scaffold
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Novel approaches for PET imaging of endometriosis

Zhang, Hongchao; Eriksson, Olof; Olovsson, Matts; Wilson, Viola et al.

Part of Nuclear Medicine and Biology, 2026

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• DOI for Novel approaches for PET imaging of endometriosis
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Toward generalizable predictive models for DNA-encoded libraries

Poongavanam, Vasanthanathan; Turunen, S Pauliina; Sandberg, Kristian; Yngve, Ulrika et al.

Part of Drug Discovery Today, 2026

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• DOI for Toward generalizable predictive models for DNA-encoded libraries
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A Diastereoselective Mizoroki-Heck Reaction for Synthesis of Spirooxindole-Based Nonnatural Amino Acids Using a Boc-Protected Amine Chiral Auxiliary

Lindman, Jens; Puthiyaparambath, Sharathna; Gising, Johan; Odell, Luke R. et al.

Part of Synlett, p. 2009-2013, 2025

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• DOI for A Diastereoselective Mizoroki-Heck Reaction for Synthesis of Spirooxindole-Based Nonnatural Amino Acids Using a Boc-Protected Amine Chiral Auxiliary
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A Multicomponent aza-Prins Strategy for the Diastereoselective Synthesis of Piperidine-Fused Dihydroquinazolinones

Dybeck, Lovisa; Baudoin, Morgane; Odell, Luke R.

Part of European Journal of Organic Chemistry, 2025

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• DOI for A Multicomponent aza-Prins Strategy for the Diastereoselective Synthesis of Piperidine-Fused Dihydroquinazolinones
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A Phase I/IIa Clinical Trial to Evaluate Safety and Adrenal Uptake of Para-Chloro-2-[¹⁸F]Fluoroethyletomidate in Healthy Volunteers and Patients with Primary Aldosteronism

Gillett, Daniel; Senanayake, Russell; MacFarlane, James; Bashari, Waiel et al.

Part of Journal of Nuclear Medicine, p. 434-440, 2025

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• DOI for A Phase I/IIa Clinical Trial to Evaluate Safety and Adrenal Uptake of Para-Chloro-2-[¹⁸F]Fluoroethyletomidate in Healthy Volunteers and Patients with Primary Aldosteronism

A preclinical study on the influence of linkers in [⁶⁸Ga]Ga-NOTA-X-RM26 radiotracers for PET imaging of GRPR expression

Olaniran Håkansson, Esther; Zelepukin, Ivan V.; Obeid, Karim; Bitzios, Athanasios et al.

Part of EJNMMI Research, 2025

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• DOI for A preclinical study on the influence of linkers in [⁶⁸Ga]Ga-NOTA-X-RM26 radiotracers for PET imaging of GRPR expression
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Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations

Beveridge, Julia; Söderström, Marcus; Balestri, Lorenzo; Prieto-Díaz, Rubén et al.

Part of Synlett, p. 2666-2670, 2025

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• DOI for Benzylhydroxamic Acids as IRAP Inhibitors: Sulfonamide Variations
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Defluorinative thio-functionalization: direct synthesis of methyl-dithioesters from trifluoromethylarenes

Söderström, Marcus; Olaniran Håkansson, Esther; Odell, Luke R.

Part of Chemical Communications, p. 145-148, 2025

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• DOI for Defluorinative thio-functionalization: direct synthesis of methyl-dithioesters from trifluoromethylarenes
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Derivatization of Small Molecules using Deuterated Analog of Reactive Matrix to Facilitate Identification in Mass Spectrometry Imaging

Vallianatou, Theodosia; Ilic Balestri, Lorenzo Jacopo; Nilsson, Anna; Zhang, Xiaoqun et al.

Part of Chemistry-Methods, 2025

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• DOI for Derivatization of Small Molecules using Deuterated Analog of Reactive Matrix to Facilitate Identification in Mass Spectrometry Imaging
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Insulin-regulated aminopeptidase inhibitor C9 restores cellular activity in methadone-damaged primary cell cultures

Stam, Frida; Lind, Sara Florén; Nylander, Erik; Olaniran Håkansson, Esther et al.

Part of Neuroscience Letters, 2025

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• DOI for Insulin-regulated aminopeptidase inhibitor C9 restores cellular activity in methadone-damaged primary cell cultures
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Novel Macrocyclic Peptidomimetics Targeting the Insulin-Regulated Aminopeptidase (IRAP): Design, Synthesis and Evaluation

Olaniran Håkansson, Esther; Balestri, Lorenzo Jacopo Ilic; Puthiyaparambath, Sharathna; Moes, Sebastian et al.

Part of RSC Medicinal chemistry, p. 5059-5069, 2025

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• DOI for Novel Macrocyclic Peptidomimetics Targeting the Insulin-Regulated Aminopeptidase (IRAP): Design, Synthesis and Evaluation
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One-pot, chemoselective desulfurative functionalization of cysteine containing peptides using pyridinium salts

van den Heuvel, Jeroen W.; Olaniran Håkansson, Esther; Skillinghaug, Bobo; Odell, Luke R.

Part of Chemical Communications, p. 10347-10350, 2025

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• DOI for One-pot, chemoselective desulfurative functionalization of cysteine containing peptides using pyridinium salts
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PET imaging of platelet derived growth factor receptor β in lung fibrosis

Wegrzyniak, Olivia; Lechi, Francesco; Rokka, Johanna; Mitran, Bogdan et al.

Part of EJNMMI Radiopharmacy and Chemistry, 2025

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• DOI for PET imaging of platelet derived growth factor receptor β in lung fibrosis
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Pretargeted brain PET imaging reveals amyloid-β pathology using a TCO-modified antibody and a fluorine-18-labeled tetrazine

Lopes van den Broek, Sara; Eriksson, Jonas; Yang, Qiaojun; Bucher, Nadja M. et al.

Part of Translational Neurodegeneration, 2025

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• DOI for Pretargeted brain PET imaging reveals amyloid-β pathology using a TCO-modified antibody and a fluorine-18-labeled tetrazine
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Reduction of negative charge in mercaptoacetyl-based chelators influences the biodistribution of prostate-specific membrane antigen-targeting pseudopeptides labeled with technetium-99m

Bezverkhniaia, Ekaterina; Kanellopoulos, Panagiotis; Rosenström, Ulrika; Tolmachev, Vladimir M. et al.

Part of ACS Pharmacology & Translational Science, p. 3600-3612, 2025

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• DOI for Reduction of negative charge in mercaptoacetyl-based chelators influences the biodistribution of prostate-specific membrane antigen-targeting pseudopeptides labeled with technetium-99m
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Repeated positron emission tomography tracing neutrophil elastase in a porcine intensive-care sepsis model

Wilske, Frida; Eriksson, Olof; Amini, Rose-Marie; Estrada, Sergio et al.

Part of Intensive Care Medicine Experimental, 2025

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• DOI for Repeated positron emission tomography tracing neutrophil elastase in a porcine intensive-care sepsis model
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Synthesis and In Vitro Profiling of Psilocin Derivatives: Improved Stability and Synthetic Properties

Eklund, Julia; Bremberg, Ulf; Larsson, Jessica; Torkelsson, Edvard et al.

Part of Journal of Medicinal Chemistry, p. 7153-7165, 2025

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• DOI for Synthesis and In Vitro Profiling of Psilocin Derivatives: Improved Stability and Synthetic Properties
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Synthesis and preclinical evaluation of gastrin releasing peptide receptor antagonist [¹⁸F]MeTz-PEG2-RM26 for positron emission tomography

Kanellopoulos, Panagiotis; Lundmark, Fanny; Abouzayed, Ayman; Balestri, Lorenzo Jacopo Ilic et al.

Part of EJNMMI Radiopharmacy and Chemistry, 2025

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• DOI for Synthesis and preclinical evaluation of gastrin releasing peptide receptor antagonist [¹⁸F]MeTz-PEG2-RM26 for positron emission tomography
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¹⁸F-labelling of nitrogen-containing aryl boronates: anti-cancer drug melflufen as a case study

Bajerke, Kevin; Lehmann, Fredrik; Antoni, Gunnar; Szabó, Kálmán J.

Part of Organic Chemistry Frontiers, p. 6411-6417, 2024

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• DOI for ¹⁸F-labelling of nitrogen-containing aryl boronates: anti-cancer drug melflufen as a case study
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[68Ga]Ga-ABY-025 PET in HER2-positive breast cancer: Benefits and pitfalls in staging of axillary disease

Alhuseinalkhudhur, Ali; Lindman, Henrik; Liss, Per; Frejd, Fredrik et al.

Part of Journal of Clinical Oncology, 2024

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• DOI for [68Ga]Ga-ABY-025 PET in HER2-positive breast cancer: Benefits and pitfalls in staging of axillary disease

Altered amyloid-β structure markedly reduces gliosis in the brain of mice harboring the Uppsala APP deletion

Pagnon de la Vega, María; Syvänen, Stina; Giedraitis, Vilmantas; Hooley, Monique et al.

Part of Acta neuropathologica communications, 2024

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• DOI for Altered amyloid-β structure markedly reduces gliosis in the brain of mice harboring the Uppsala APP deletion
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Benzylhydroxamic acids as inhibitors of insulin regulated aminopeptidase (IRAP)

Beveridge, Julia; Söderström, Marcus; Prieto-Díaz, Rubén; Gutierrez-de-Teran, Hugo et al.

Part of European Journal of Medicinal Chemistry Reports, 2024

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• DOI for Benzylhydroxamic acids as inhibitors of insulin regulated aminopeptidase (IRAP)
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Identification of novel and potent inhibitors of SARS-CoV-2 main protease from DNA-encoded chemical libraries

Akaberi, Dario; Pourghasemi, Monireh; Krambrich, Janina; Berger, Julia et al.

Part of Antimicrobial Agents and Chemotherapy, p. 1-18, 2024

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• DOI for Identification of novel and potent inhibitors of SARS-CoV-2 main protease from DNA-encoded chemical libraries
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Inhibition of Insulin-Regulated Aminopeptidase by Imidazo[1,5-α]pyridines; Synthesis and Evaluation

Engen, Karin; Lundbäck, Thomas; Yadav, Anubha; Puthiyaparambath, Sharathna et al.

Part of International Journal of Molecular Sciences, 2024

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• DOI for Inhibition of Insulin-Regulated Aminopeptidase by Imidazo[1,5-α]pyridines; Synthesis and Evaluation
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N-(Heteroaryl)thiophene sulfonamides as angiotensin AT2 receptor ligands

Wannberg, Johan; Gising, Johan; Henriksson, Martin; Vo, Duc Duy et al.

Part of European Journal of Medicinal Chemistry, 2024

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• DOI for N-(Heteroaryl)thiophene sulfonamides as angiotensin AT2 receptor ligands
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Optimized method for fluorine-18 radiolabeling of Affibody molecules using RESCA

Lechi, Francesco; Eriksson, Jonas; Odell, Luke R.; Wegrzyniak, Olivia et al.

Part of EJNMMI Radiopharmacy and Chemistry, 2024

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• DOI for Optimized method for fluorine-18 radiolabeling of Affibody molecules using RESCA
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PET imaging of GABA_A receptors in pancreatic islets by [¹¹C]flumazenil

Maloum-Rami, Faïza; Cheung, Pierre; Antoni, Gunnar; Jin, Zhe et al.

Part of EJNMMI Research, 2024

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• DOI for PET imaging of GABA_A receptors in pancreatic islets by [¹¹C]flumazenil
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PET tracers beyond [18F]FDG: Chapter 5: [11C]PE2I & [18F]FE-PE2I

Crnic Bojkovic, Tea; Sigfridsson, Jonathan; Stepanov, Vladimir; Eriksson, Jonas et al.

Part of EANM Technologists’ Guide, 2024

Article, review/survey

• DOI for PET tracers beyond [18F]FDG: Chapter 5: [11C]PE2I & [18F]FE-PE2I

Radiation dosimetry of para-chloro-2-[¹⁸F]fluoroethyl-etomidate: a PET tracer for adrenocortical imaging

Silins, Isabella; Moreno, Adrian; Wall, Anders; Aigbirhio, Franklin et al.

Part of EJNMMI Research, 2024

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• DOI for Radiation dosimetry of para-chloro-2-[¹⁸F]fluoroethyl-etomidate: a PET tracer for adrenocortical imaging
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Reduction of renal activity retention of radiolabeled albumin binding domain-derived affinity proteins using a non-residualizing label strategy compared with a cleavable glycine-leucine-glycine-lysine-linker

Lundmark, Fanny; Vorobyeva, Anzhelika; Liu, Yongsheng; Lindbo, Sarah et al.

Part of Molecular Medicine Reports, 2024

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• DOI for Reduction of renal activity retention of radiolabeled albumin binding domain-derived affinity proteins using a non-residualizing label strategy compared with a cleavable glycine-leucine-glycine-lysine-linker
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Regional distribution of mechanical strain and macrophage-associated lung inflammation after ventilator-induced lung injury: an experimental study

Liggieri, Francesco; Chiodaroli, Elena; Pellegrini, Mariangela; Puuvuori, Emmi et al.

Part of Intensive Care Medicine Experimental, 2024

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• DOI for Regional distribution of mechanical strain and macrophage-associated lung inflammation after ventilator-induced lung injury: an experimental study
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Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET

Schlein, Eva; Rokka, Johanna; Odell, Luke R.; Lopes van den Broek, Sara et al.

Part of EJNMMI Radiopharmacy and Chemistry, 2024

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• DOI for Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
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Synthesis of N-Alkenylated Heterocycles via T₃P-Promoted Condensation with Ketones

Balestri, Lorenzo Jacopo Ilic; Beveridge, Julia; Gising, Johan; Odell, Luke R.

Part of Journal of Organic Chemistry, p. 11203-11214, 2024

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• DOI for Synthesis of N-Alkenylated Heterocycles via T₃P-Promoted Condensation with Ketones
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The decanoate esters of nandrolone, testosterone, and trenbolone induce steroid specific memory impairment and somatic effects in the male rat

Zelleroth, Sofia; Stam, Frida; Nylander, Erik; Ellinor, Kjellgren et al.

Part of Hormones and Behavior, 2024

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• DOI for The decanoate esters of nandrolone, testosterone, and trenbolone induce steroid specific memory impairment and somatic effects in the male rat
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The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds

Gising, Johan; Honarnejad, Saman; Bras, Maaike; Baillie, Gemma L. et al.

Part of International Journal of Molecular Sciences, 2024

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• DOI for The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds
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Two Novel [⁶⁸Ga]Ga-Labeled Radiotracers Based on Metabolically Stable [Sar¹¹]RM26 Antagonistic Peptide for Diagnostic Positron Emission Tomography Imaging of GRPR-Positive Prostate Cancer

Kanellopoulos, Panagiotis; Bezverkhniaia, Ekaterina; Abouzayed, Ayman; Rosenström, Ulrika et al.

Part of ACS Omega, p. 18608-18616, 2024

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• DOI for Two Novel [⁶⁸Ga]Ga-Labeled Radiotracers Based on Metabolically Stable [Sar¹¹]RM26 Antagonistic Peptide for Diagnostic Positron Emission Tomography Imaging of GRPR-Positive Prostate Cancer
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¹⁷⁷Lu-labeled PSMA targeting therapeutic with optimized linker for treatment of disseminated prostate cancer; evaluation of biodistribution and dosimetry

Abouzayed, Ayman; Seitova, Kamila; Lundmark, Fanny; Bodenko, Vitalina et al.

Part of Frontiers in Oncology, 2023

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• DOI for ¹⁷⁷Lu-labeled PSMA targeting therapeutic with optimized linker for treatment of disseminated prostate cancer; evaluation of biodistribution and dosimetry
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[¹⁸F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44

Cheung, Pierre; Amin, Mohammad A.; Zhang, Bo; Lechi, Francesco et al.

Part of Pharmaceutics, 2023

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• DOI for [¹⁸F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44
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A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane

Schembri, Luke S; Olaniran, Esther; Söderström, Marcus; Skillinghaug, Bobo et al.

Part of Advanced Synthesis and Catalysis, p. 1839-1845, 2023

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• DOI for A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane
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Acute nicotine exposure blocks aromatase in the limbic brain of healthy women: A [11C]cetrozole PET study

Dubol, Manon; Immenschuh, Jana; Jonasson, My; Takahashi, Kayo et al.

Part of Comprehensive Psychiatry, 2023

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• DOI for Acute nicotine exposure blocks aromatase in the limbic brain of healthy women: A [11C]cetrozole PET study
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Acyl Amidines by Pd-Catalyzed Aminocarbonylation: One-Pot Cyclizations and ¹¹C Labeling

Rydfjord, Jonas; Roslin, Sara; Roy, Tamal; Abbas, Alaa et al.

Part of Journal of Organic Chemistry, p. 5078-5089, 2023

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• DOI for Acyl Amidines by Pd-Catalyzed Aminocarbonylation: One-Pot Cyclizations and ¹¹C Labeling
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First-in-human evaluation of [¹⁸F]CETO: a novel tracer for adrenocortical tumours

Silins, Isabella; Sundin, Anders; Lubberink, Mark; O'Sullivan, Lleah et al.

Part of European Journal of Nuclear Medicine and Molecular Imaging, p. 398-409, 2023

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• DOI for First-in-human evaluation of [¹⁸F]CETO: a novel tracer for adrenocortical tumours
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In Vivo Visualization and Quantification of Neutrophil Elastase in Lungs of COVID-19 Patients: A First-in-Humans PET Study with ¹¹C-NES

Antoni, Gunnar; Lubberink, Mark; Sörensen, Jens; Lindström, Elin et al.

Part of Journal of Nuclear Medicine, p. 145-148, 2023

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• DOI for In Vivo Visualization and Quantification of Neutrophil Elastase in Lungs of COVID-19 Patients: A First-in-Humans PET Study with ¹¹C-NES
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